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1-methyl-4-[4-(4-phenylpyrimidin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
N-ethyl-2-methyl-6-(piperidin-4-yl)-N-propylpyrimidin-4-amine
4-(2,1,3-benzoxadiazol-4-yl)-1-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-methyl-2-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1-oxaspiro[4.5]decane-4-carboxamide
1-[4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]pyrrolidin-2-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
1-cyclopentyl-4-oxo-N3-[2-(4-phenylpiperidin-1-yl)ethyl]-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
7-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(1R,5S,8S)-8-methoxy-3-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.2.1]octane
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidin-2-amine
(1R,5R)-3-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-[4-(1,3-benzothiazol-2-yl)-1,4-diazepane-1-carbonyl]-2-methylpyrimidin-4-ol
(furan-3-ylmethyl)(methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
1-{[3-(cyclopentyloxy)phenyl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-[2-(2-fluorophenoxy)ethyl]-1-(2-methoxyethyl)-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
6-(2-methoxyphenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyridazin-3-amine
(3aS,7aR)-2-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
8-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(benzyloxy)piperidin-1-yl]ethan-1-one
5-{[ethyl(oxolan-2-ylmethyl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-({[2-(4-chloro-1H-pyrazol-1-yl)ethyl]amino}methyl)pyrrolidin-3-ol
N-(1H-imidazol-2-ylmethyl)-1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2-hydroxyethyl)-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[1-(4-methanesulfonylphenyl)ethyl]propanamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidine
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-benzyl-1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine-4-carboxamide
6-ethyl-2-methyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}quinoline
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}thiomorpholine
1-[(3-fluorophenyl)methyl]-4-[(propan-2-yl)amino]pyrrolidin-2-one
1-[(2S,4R)-1-[(2,4-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
ethyl 2-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}amino)acetate
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]cyclopropanecarboxamide
1-(2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl)pyrrolidine
2-(pyridin-3-yl)-N-[1-(thiophen-3-yl)propan-2-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-(2,3-difluoro-4-methoxybenzoyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-[2-(3-methoxyphenyl)ethyl]piperidine
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2,2-dimethylpropan-1-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
3-(2-methoxyethyl)-1-[(2-methylphenyl)methyl]-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-[2-(2-fluoro-4-methoxyphenyl)-1H-imidazol-1-yl]-3-(pyrrolidin-1-yl)propan-2-ol
N-[(1S,2R)-2-aminocyclobutyl]-1-phenylmethanesulfonamide
2-(2-aminoethyl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}quinazolin-4-amine
1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyridin-3-yl)ethan-1-one
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-(thiophen-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
[1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-3-yl]methanamine