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N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-(aminomethyl)-2-(3-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
dimethyl({[(1R,5S,6S)-3-{[2-(trifluoromethyl)phenyl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
(3R,4R)-3-cyclopropyl-4-methyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-ol
3-(5-{[2-(benzyloxy)phenyl]methyl}-1,2,4-oxadiazol-3-yl)pyridazine
1-(2-{[(8-chloro-4-hydroxyquinolin-2-yl)methyl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N-(5-chloro-2-methylphenyl)-7-(3-methoxypropyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
5-(1-cyclobutylpyrrolidin-2-yl)-N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}thiophene-2-carboxamide
2-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
1-{3-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}azepan-2-one
1,3-dimethyl-6-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-9-methyl-3,9-diazaspiro[5.6]dodecane
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)propanamide
N-(oxan-3-yl)-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
4-{2-[(4-benzyl-5-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}morpholine
(3R,9R)-11-(naphthalene-1-carbonyl)-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
2-hydroxy-4-(methylsulfanyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
N-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
8-[4-(dimethylamino)butan-2-yl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-({3-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidine-4-carbonitrile
2-{1-[1-(5-fluoro-3,8-dimethylquinolin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
5-cyclopropyl-N-(2,2-dimethyloxan-4-yl)-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(azepan-1-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
6-(2-chlorophenyl)-2-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
(3-{3-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}propyl)dimethylamine
2-(4-chlorophenoxy)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
[(3R,4R)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]-1-(2-fluorophenyl)ethan-1-ol
4-hydroxy-N-{3-[methyl(phenyl)amino]propyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N,1-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-indole-6-carboxamide
3-chloro-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
(1S,5R)-3-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3R,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
3-benzyl-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-diethyl-1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
1-(1-cyclopropylethyl)-5-(3,5-difluorophenyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(2,3-dihydro-1H-inden-2-yl)-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
[(5-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
2-(3-methylbutyl)-8-(4-methylpiperazine-1-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-{[4-methyl-5-(1-propylpiperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
N-(2-phenylethyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
3-[5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenol
4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1,3-dimethylpiperazin-2-one
1-[(2S)-2-methoxy-2-phenylacetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4S)-4-(4-{[(3-methoxyphenyl)formamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide