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6-methoxy-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidin-4-amine
(2R)-2-[(2-amino-5-ethylpyrimidin-4-yl)amino]-3-phenylpropan-1-ol
1-(3-cyanophenyl)-3-[2-(4-ethylmorpholin-2-yl)ethyl]urea
2-(2-{1-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}phenoxy)ethan-1-ol
1-(2-chlorophenyl)-3-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
[2-(dimethylamino)ethyl](methyl)(2-{[4-(trifluoromethyl)pyrimidin-2-yl]oxy}hex-5-en-1-yl)amine
(1R,9aR)-1-[({[1-(hydroxymethyl)cyclopentyl]methyl}(methyl)amino)methyl]-octahydro-1H-quinolizin-1-ol
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-5-(propan-2-yl)pyrimidine
3-[1-(dimethylsulfamoyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
4-(4-chlorophenyl)-1-(3-hydroxypyrrolidin-1-yl)butan-1-one
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(2-cyclopentylacetyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[2-(2-butoxy-4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-3-ol
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]piperazine-1-carboxamide
1-(2-cyclopropyl-4-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-hydroxyethan-1-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
4-methyl-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}thiophene-2-sulfonamide
N-({1-[(4,5-dimethylfuran-2-yl)methyl]pyrrolidin-3-yl}methyl)-2-(morpholin-4-yl)-2-oxoacetamide
1-(furan-2-ylmethyl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2,2,2-trifluoroethyl)acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3-carboxamide
2-[4-(pentan-3-yl)piperazin-1-yl]-5-propylpyrimidine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
2-methoxy-N-{3-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]phenyl}acetamide
N-[(3R)-1-benzylpyrrolidin-3-yl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
3-[2-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-pyrrol-1-yl]pyridine
5-ethyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[1-(3,4-difluorobenzenesulfonyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-(2-ethylpyrimidine-5-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
{2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}urea
3-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4,7-trimethyl-1H-indole-2-carboxamide
2,2-dimethyl-1-[4-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperazin-1-yl]propan-1-one
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
N-[3-(1H-imidazol-1-yl)butyl]-2,6-dimethylquinoline-4-carboxamide
methyl 9-{methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}-3-azaspiro[5.5]undecane-3-carboxylate
2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-[4-(propan-2-yl)phenyl]acetic acid
(3aS,6aS)-2-methyl-5-[2-(morpholin-4-yl)pyridine-3-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-{3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenoxy}acetamide
5-fluoro-N,N-dimethyl-2-[3-(pyrimidin-4-yl)piperidin-1-yl]pyrimidin-4-amine
2-(3,5-difluorophenyl)-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]acetamide
2-methoxy-1-{4-[4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
1-(6-chloropyridazin-3-yl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-amine
2-{[5-(5-chlorothiophen-2-yl)-4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-(3,4-dimethylphenyl)-2-{[3-(pyridin-4-yl)propyl]amino}acetamide
N-[(1-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}piperidin-3-yl)methyl]acetamide