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[(3R,4R)-4-[(dimethylamino)methyl]-1-(3-phenyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-{[3-(1H-imidazol-1-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(8-methoxyquinolin-5-yl)methyl]-N,3-dimethyl-1,2-oxazole-5-carboxamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-1,4-diazepane-6-carboxylic acid
(4aS,8aR)-6-[3-(furan-2-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
2-(2,5-dimethoxyphenyl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-methyl-2-oxo-8-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(5S,9aS,9bS)-5-[3-(ethoxymethyl)-4-methoxyphenyl]-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(4-fluorophenoxymethyl)piperidine
3-(2-methoxyphenoxy)-1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}azetidine
1-(3-methoxypropyl)-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
1-{[5-(4-methyl-1H-imidazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}azocane
2-{[(1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)oxy]methyl}pyridine
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(piperidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
2-fluoro-N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
{3-[(3-chlorophenyl)methyl]-1-[(6-fluoroquinolin-2-yl)methyl]piperidin-3-yl}methanol
1-[3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-oxopropyl]azepan-2-one
5-(1-ethyl-1H-pyrazole-4-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-(1-phenylcyclopropanecarbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
7-(2-methoxyethyl)-2-[(2-methyl-1-benzothiophen-3-yl)methyl]-2,7-diazaspiro[4.5]decane
6-(benzyloxy)-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-3-(2-fluorophenyl)-3-phenylpropanamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-3-yl]methanol
5-methyl-N-[2-(6-methylpyridin-2-yl)ethyl]-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
5-(5-fluoropyridin-2-yl)-1,2,3,4-tetrahydroisoquinoline
N,2,3,5,6-pentamethyl-N-(prop-2-en-1-yl)benzamide
1'-(5-fluoropyridine-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]oxane-4-carboxamide
3-{[(1,5-dimethyl-1H-pyrazol-3-yl)methyl](methyl)amino}-1-phenylpropan-1-ol
1-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-4-yl}-2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
1-(2-methylpyridin-4-yl)-4-{[5-(oxan-2-yl)furan-2-yl]methyl}-1,4-diazepane
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
[(2,2-dimethyloxan-4-yl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
2-benzyl-8-(2-hydroxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-1-(morpholine-4-sulfonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
{[(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
[(3R,4R)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
5-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2-methylphenol
N-[(1-cyclopentylpiperidin-4-yl)methyl]-6-oxo-N-(oxolan-2-ylmethyl)-1,6-dihydropyridine-2-carboxamide
(3S,4R)-1-(3-ethoxypropanoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-(oxolan-2-ylmethyl)-4-[4-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)piperidin-3-ol
2-{[(3-ethoxyphenyl)methyl][(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}ethan-1-ol
2-[4-(4-aminopyrimidin-2-yl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol