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2-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
3-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
N3-(3-methylbutyl)-N5-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
5-cyclopropyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-phenylpiperazin-2-one
4,4-difluoro-N-(2-fluoro-4-methoxyphenyl)piperidine-1-carboxamide
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[4-(pyrimidin-5-yl)phenyl]methanesulfonamide
{4-[(3-chloro-4-fluorophenyl)methyl]-1-methylpiperazin-2-yl}methanol
8-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]acetyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,3-dimethylphenyl)-N-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(4aS,8aR)-6-[(3-methoxyphenyl)methyl]-1-methyl-decahydro-1,6-naphthyridine-4a-carboxylic acid
(3S,4R)-1-[2-(dimethylamino)benzoyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-methyl-6-[1-(thiophen-3-ylmethyl)piperidin-3-yl]pyrimidin-4-ol
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(morpholin-4-yl)ethan-1-one
2-{1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]pyrrolidin-2-yl}pyridine
2-[3-(piperazin-1-ylmethyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
2-[(1-{1,9-dioxaspiro[5.5]undecan-4-yl}piperidin-4-yl)oxy]pyrimidine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylacetamide
(1R,5S)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonane
2-methyl-6-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
N-(2-{1-[2-(ethylsulfanyl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)piperidine-1-carboxamide
(3S,4S)-N-(2,5-di-tert-butylphenyl)-3,4-bis(hydroxymethyl)pyrrolidine-1-carboxamide
4-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
1-{3-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
N-methyl-N-(thiophen-3-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-methyl-5-oxopyrrolidin-1-yl)acetamide
N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-[3-(2-methoxyphenyl)propyl]-2-(2-oxopiperidin-1-yl)acetamide
2-({[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}amino)acetamide
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
[(2-chloro-4-fluorophenyl)methyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
1-{1'-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
5-methyl-3-(2,4,6-trimethylphenyl)pyridin-2-amine
N-{3-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}acetamide
N-methyl-2-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}acetamide
2-methyl-6-(piperidin-3-yl)-N-{[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-4-amine
2-(adamantan-1-yl)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]ethan-1-one
2-ethyl-8-(2-hydroxynaphthalene-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
9-(3-ethyl-1,2-oxazole-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-1-[(4-chlorophenyl)methyl]-N-(cyclopropylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
{[(2R,5S)-5-(2H-1,3-benzodioxol-5-ylmethyl)oxolan-2-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
3-(butan-2-yl)-5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-ethyl-N-(1,2-oxazol-3-ylmethyl)-1H-indole-5-carboxamide
4-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-dimethyl-1H-pyrazole
(3S,4R)-1-[2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(pyridine-3-carbonyl)pyrrolidine-3-carboxylic acid