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N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-4-(piperidin-1-ylmethyl)benzamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(2-hydroxyphenyl)methyl]-N-methylbenzamide
1-(4-chlorophenyl)-N-{[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
3-[1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-(azepan-1-yl)-2-(4-hydroxyphenyl)acetic acid
3-[1-(quinoxaline-6-carbonyl)piperidin-3-yl]benzoic acid
N,1-dimethyl-6-propyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-ethyl-2-{4-[4-(thiophen-2-yl)-1H-imidazol-1-yl]phenyl}acetamide
5-tert-butyl-4-({8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)furan-2-carboxamide
(3S,4R)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-(acetamidomethyl)-N-(trimethyl-1H-pyrazol-4-yl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-methoxypropanamide
({5-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]thiophen-3-yl}methyl)dimethylamine
N-(3-hydroxypropyl)-1-[1-(naphthalen-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
3-(3-fluorophenyl)-1-methyl-3-(2-oxo-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethyl)pyrrolidine-2,5-dione
ethyl 2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetate
2-methoxy-5-{1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
3-(2-methoxyethyl)-1-{[(2-phenylethyl)carbamoyl]methyl}piperidine-3-carboxylic acid
4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-N-methylpyridin-2-amine
2-methyl-5-{4-[3-(pyridin-3-yl)propanoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[3-(morpholin-4-yl)propyl]benzamide
N-(1-carbamoylcyclopentyl)-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-(2-amino-5,6-dimethylpyrimidin-4-yl)-4-benzylpiperidin-4-ol
methyl 2-(4-{[1-(2,3-dimethylphenyl)piperidin-4-yl]amino}piperidin-1-yl)acetate
5-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-N-(propan-2-yl)pyrimidin-2-amine
2,5,7-trimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-N-(2,2-difluoroethyl)benzene-1-sulfonamide
4-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-methyl-2-phenylpiperazine
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
N-cyclohexyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
7-(3-methoxyphenyl)-2-(3-methyl-1H-pyrazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-propyl-6-{pyrazolo[1,5-a]pyridin-3-yl}-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
(3R,4R)-3-cyclobutyl-4-methyl-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-ol
1-ethyl-4-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}piperazine-2,3-dione
N-[2-(1,2,5-thiadiazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
5-fluoro-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,2-dimethyloxane-4-carboxamide
2-(1-{[1-(quinoxaline-6-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
2-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-ol
2-(4-chloro-1H-pyrazole-3-carbonyl)-8-methyl-2,8-diazaspiro[4.5]decane
1-{[bis(prop-2-en-1-yl)carbamoyl]methyl}piperidine-3-carboxamide
4-(2H-1,3-benzodioxol-5-yl)-2-[5-(furan-2-yl)-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-(thiophen-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(3R,4S)-1-[3-(3-fluorophenyl)propanoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
7-(2-methylphenyl)-4-[5-(propan-2-yl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole