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3-(2H-1,3-benzodioxol-5-yl)-1-{3-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}propan-1-one
1-ethyl-N-methyl-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-4-carboxamide
1-methanesulfonyl-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-(3-acetylphenyl)-4-{[(2S,5R)-2,5-dimethylpiperazin-1-yl]methyl}benzamide
ethyl 2-[methyl(3-oxo-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl)amino]acetate
N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-2-methylphenol
3-fluoro-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}benzamide
5-(1-ethyl-1H-imidazol-5-yl)-1-[4-(oxolan-2-yl)butyl]-4-phenyl-1H-imidazole
N-benzyl-4-cyclopentyl-3-oxopiperazine-1-sulfonamide
6-(pyridin-3-yl)-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
3,5-dimethoxy-2-{[3-(methylcarbamoyl)piperidin-1-yl]methyl}benzoic acid
N-(1-benzothiophen-2-ylmethyl)-4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methylpyrimidin-2-amine
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-(propan-2-yloxy)propan-1-one
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-{[(3,5-dimethoxyphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-acetyl-N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
N-benzyl-4-hydroxy-2-methyl-N-(2-phenylethyl)pyrimidine-5-carboxamide
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
(3aR,6aR)-2-(2-chloro-6-methylbenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]-3-(methylsulfanyl)propan-1-one
1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-({6-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrazin-2-yl}sulfanyl)acetic acid
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)amine
N-(butan-2-yl)-3-methyl-N-(pyridin-4-ylmethyl)furan-2-carboxamide
methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
1-benzyl-4-({4-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazine
N-methyl-1-[1-(2-phenylethyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-3-carboxamide
3-(propan-2-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-pyrazole-5-carboxamide
N3-[1-(6-methoxynaphthalen-2-yl)ethyl]-N5-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-ethyl-N-[3-(furan-2-yl)-3-phenylpropyl]pyrimidine-5-carboxamide
2-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
3-[(3-hydroxypiperidin-1-yl)sulfonyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
ethyl 1-(5-methyl-1H-pyrazole-3-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
7-[(2,3-dimethoxyphenyl)methyl]-2-(3-methylbutanoyl)-2,7-diazaspiro[4.5]decan-6-one
3-butyl-4-(2-methoxybenzenesulfonyl)-1-methylpiperazin-2-one
1-[({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)carbamoyl)methyl]piperidine-4-carboxamide
N-ethyl-5-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyrimidin-2-amine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]piperidin-4-ol
4-methoxy-N-{[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(2,4-difluorophenyl)ethan-1-one
N-(3-chloro-4-methoxyphenyl)-6-[2-(phenylsulfanyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
3-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1H-pyrazol-5-amine
3-cyclopentyl-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
6-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]pyrazine-2-carboxamide
8-[(3-ethoxy-4-hydroxyphenyl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-methyl-1-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-dihydroisoquinoline-4-carboxamide