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1-{[1-(6-methylpyridazin-3-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
ethyl 2-({1-[3-(4-fluorobenzenesulfonamido)phenyl]piperidin-4-yl}(methyl)amino)acetate
methyl({[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
8-methoxy-3-(quinolin-6-ylmethyl)-3,4-dihydroquinazolin-4-one
8-acetyl-2-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5,6-dimethyl-N-[1-(pyrazin-2-yl)piperidin-3-yl]pyrimidin-4-amine
1-methyl-5-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
2-(1-cyclopentyl-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl)ethan-1-ol
N-[(3S,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyridine-4-carboxamide
2-[4-(thiomorpholine-4-sulfonyl)phenyl]pyridine-4-carboxamide
4-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-methoxypyridine-3-carbonitrile
2-{4-[4-fluoro-2-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}-N-methylacetamide
1-(furan-2-ylmethyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}piperidine-3-carboxamide
8-(3-fluoropyridin-4-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-[4-(thiomorpholine-4-sulfonyl)phenyl]quinazolin-4-amine
[(5-chloro-2,3-dimethoxyphenyl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-(cyclopropylmethyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4-methylphenol
6-methoxy-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]pyrimidin-4-amine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,4-dimethoxybenzamide
N-{2-[1-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)piperidin-2-yl]ethyl}acetamide
4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)morpholine
2-[1-cyclopentyl-4-(2,3-dimethylquinoxaline-6-carbonyl)piperazin-2-yl]ethan-1-ol
2-cyclopropyl-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-methyl-5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-methyl-5-propyl-N-[3-(pyrrolidin-1-yl)propyl]-1,3,4-oxadiazol-2-amine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
2-ethyl-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]pyrimidine-5-carboxamide
[(4aS,8aR)-6-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
14-[5-(3-chlorophenyl)furan-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-methyl-3-phenyl-8-(pyridine-4-carbonyl)-1,8-diazaspiro[4.5]decane
1-[4-(benzenesulfonyl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
1-[(5-propylfuran-2-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-(2-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}quinolin-6-yl)acetamide
methyl 6-[(diethylamino)methyl]-3-(furan-2-amido)thieno[2,3-b]pyridine-2-carboxylate
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
2-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
5-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
5-ethyl-4-[4-(morpholin-4-yl)piperidin-1-yl]pyrimidin-2-amine
N-butyl-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
4-methoxy-N-methyl-3-[3-(methylsulfanyl)phenyl]benzamide
N-(2,4-dimethoxyphenyl)-3-(morpholin-4-yl)piperidine-1-carboxamide
N-[(2S)-1-cyclohexyl-3-hydroxypropan-2-yl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
[1-(5-{[3-(methylsulfanyl)propyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol