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7-fluoro-2-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}quinoline-4-carboxamide
4-[2-(1H-imidazol-2-yl)benzoyl]-2-(4-methylpentyl)morpholine
3-(cyclopropylmethyl)-1-[3-(methylsulfanyl)propanoyl]piperidine-3-carboxylic acid
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
3-chloro-4-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)formamido]acetic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(2-hydroxyethyl)(methyl)sulfamoyl]benzamide
4-{1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}pyridine
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}oxane-2-carboxamide
3-(5-{2-[(1-phenylethyl)carbamoyl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
1-(4-methoxyphenyl)-3-methyl-4-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)piperazin-2-one
1-methyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
3-(2,6-dimethoxyphenyl)-5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazole
3-{[4-(3-hydroxyphenyl)piperidin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
ethyl 5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
5-chloro-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
2-oxo-3-(pentan-3-yl)-1-(pyrrolidin-3-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(1H-indol-3-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carboxylic acid
2-benzyl-N-(4-ethoxy-2-fluorophenyl)-3-oxopiperazine-1-carboxamide
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-5-methylthiophene-2-carboxamide
2-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanamide
4-{5-[4-(piperidin-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl}pyridine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]pyridazine-3-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
1-[1'-(3-hydroxy-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(4-hydroxypiperidin-1-yl)acetamide
N-[(1R,3R)-3-aminocyclopentyl]-2,6-dimethoxypyridine-3-carboxamide
(2E)-1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-3-(furan-2-yl)prop-2-en-1-one
3-(2-phenoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{5-[(dimethylamino)methyl]-1,2,4-oxadiazol-3-yl}phenyl)ethan-1-ol
2-(3-phenylpropyl)-4-(thiophene-2-carbonyl)morpholine
1-(2,3-difluoro-6-methoxybenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
[(3R,4S)-1-[(3-chloro-2,4-difluorophenyl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
8-(3-hydroxypropyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(cyclohexylmethyl)(methyl)({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
3-[4-phenyl-5-(quinolin-3-yl)-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
1-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}piperidin-2-one
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-6-(propan-2-yl)pyrimidin-4-amine
7-[(3-methoxyphenyl)methyl]-2-(1-methylcyclopropanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-methoxy-8-(6-methylhept-5-en-2-yl)-1,8-diazaspiro[4.5]decan-2-one
5-{[2-(aminomethyl)morpholin-4-yl]methyl}-N-benzylpyrimidin-2-amine
4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl]pyridine
1'-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide