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5-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
6-(2-methoxyphenyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyridazin-3-amine
1-[(2-chlorophenyl)methyl]-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1,3-dimethyl-6-[4-(9H-purin-6-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
(4aR,8aR)-2-cyclopentanecarbonyl-7-(1H-imidazol-2-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
N3-benzyl-N5-[1-(furan-2-yl)ethyl]-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{2-oxo-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]ethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-(3-chloro-2-methylphenyl)-N'-[3-(pyridin-3-yloxy)propyl]propanediamide
2-[benzyl(methyl)amino]-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
2-[(3,5-dimethoxyphenyl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
2-(2-ethoxy-3-methoxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(4-methanesulfonylphenyl)methyl]-4,4-dimethylpyrrolidin-2-one
3-{1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-6-(thiophen-3-yl)pyridine-3-carboxamide
N-[1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-4-(1H-pyrazol-3-yl)benzamide
2-{1-methyl-4-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperazin-2-yl}ethan-1-ol
(1S,5R)-3-[2-(pyridin-2-ylsulfanyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{4-[(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)sulfonyl]phenyl}acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-(1H-imidazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-4-yl}methanesulfonamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-dimethylquinoline-4-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)amine
N,5-dimethyl-N-[3-(oxolan-2-yl)propyl]-1H-indazole-3-carboxamide
3-[3-oxo-4-(2-phenylethyl)piperazine-1-carbonyl]piperidine-1-carboxamide
7-fluoro-3-[({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1,2-dihydroquinolin-2-one
2-methyl-N-({methyl[1-(2-phenylethyl)piperidin-3-yl]carbamoyl}methyl)propanamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3,4,5-trimethoxybenzamide
4-[3-(3-methyl-3-phenylpiperidine-1-carbonyl)phenyl]morpholine
7-(1,3-benzothiazol-2-yl)-4-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(5-acetylthiophene-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-fluorophenyl)-3-[(oxan-3-yl)sulfamoyl]benzamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
methyl 4-[(3-benzoylpiperidin-1-yl)methyl]thiophene-2-carboxylate
2-methyl-8-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-4-{[(2,4-difluorophenyl)methyl]amino}-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-ethyl-N,5-dimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-3-carboxamide
N-cyclopropyl-4-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}pyridine-2-carboxamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,3-thiazol-2-yl)piperidine
1-[2-methoxy-5-({[3-(propan-2-yloxy)propyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
9-[1-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
7-(pyridin-3-yl)-4-(1H-pyrrole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3,4-dichlorophenyl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]morpholine
4-(4-chlorophenyl)-1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
N-{1-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
(2R,6R)-4-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
9-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one