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3-(5-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-(2-methylphenyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
3-(2-chlorophenyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-hydroxyphenyl)-N-methylpropanamide
2,6-dihydroxy-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
14-(2-fluoro-5-methylphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidine-1-carbonyl]-7-fluoro-1,2-dihydroquinolin-2-one
3-(2-{[5-(furan-3-yl)-4-(4-methylphenyl)pyrimidin-2-yl]amino}ethyl)-1,3-oxazolidin-2-one
2-cyclobutyl-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]ethan-1-one
(1R,3S)-7-(2,6-difluoro-3-methoxybenzoyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-(2-methylpropyl)pyrrolidin-2-one
(1R,2S,6R,7S)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
N-ethyl-1-(2-methylpropyl)-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(1,3-benzoxazol-2-yl)-N-[1-(4-methylpyridin-2-yl)propyl]acetamide
2-amino-4-(pyridin-3-yl)-6-[3-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}butanamide
N-(1-methyl-1H-imidazol-2-yl)-4-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}benzamide
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
ethyl N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
N-(oxolan-2-ylmethyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-4,5,6,7-tetrahydro-1-benzofuran-4-one
4-[4-(2-ethyl-1H-imidazol-1-yl)phenyl]phenol
3-{[1-(cyclohex-1-en-1-yl)ethyl]amino}-N-cyclohexylpropanamide
benzyl(ethyl){[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
(4aS,7aR)-1-(2-cyclopropylacetyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)sulfonyl]azetidin-3-yl}pyridine
5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-[phenyl(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
3-[4-(2-amino-6-methylpyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]pyrazine-2-carbonitrile
(1S,5R)-3-cyclobutanecarbonyl-6-[3-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
5-methoxy-2-{[9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N-{2-[(benzylsulfamoyl)amino]ethyl}acetamide
1,5-dimethyl-4-{1-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-(4-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)acetamide
N-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[2-(3-fluorophenyl)ethyl]-5-[4-(4-hydroxybutyl)piperazine-1-carbonyl]piperidin-2-one
2-{[4-(2-amino-6-methylpyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
1-{2-[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5R)-6-[2-(5-acetylthiophen-3-yl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3R,4R)-4-(hydroxymethyl)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperidin-3-ol
3-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]phenyl}oxolane-3-carboxamide
1-cyclopropyl-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H-pyrrole-2-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
2-{4-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]-3,5-dimethyl-1H-pyrazol-1-yl}ethan-1-ol
[(3-chloro-4-ethoxyphenyl)methyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(3-fluorophenyl)ethan-1-one
(3-{[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
5-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N'-cycloheptyl-N-[3-(pyridin-3-yloxy)propyl]butanediamide
5-methanesulfonyl-4-(piperidin-3-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine