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2-[(4-chlorophenyl)methyl]-8-(propane-1-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
5-{[(3S)-3-ethylmorpholin-4-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 4-(6-methoxypyridin-3-yl)-2-(methylsulfanyl)pyrimidine-5-carboxylate
8-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
1-[2-methoxy-5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(2-fluorobenzoyl)piperidin-3-yl]propan-1-one
5-chloro-2-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-(1,3-dimethyl-1H-pyrazol-4-yl)-4-{[(pyridin-3-yl)carbamoyl]methyl}piperazine-1-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
4-[2,2-dimethyl-3-(3-phenoxyazetidin-1-yl)propyl]morpholine
4-[(4-methoxyphenyl)methyl]-3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-1-(4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1,4-diazepan-1-yl)ethan-1-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-phenylpropanamide
1-{1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
2-{4-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}ethan-1-ol
(2S,4R)-4-amino-N-methyl-1-[2-methyl-5-(1H-pyrazol-1-yl)benzenesulfonyl]pyrrolidine-2-carboxamide
1-(2-ethylphenyl)-3-[1-(methoxymethyl)cyclopentyl]urea
1-{1-[2-(pyrazin-2-yl)acetyl]piperidin-4-yl}pyrrolidin-2-one
N-[2-(dimethylamino)ethyl]-4-(quinolin-5-yloxy)piperidine-4-carboxamide
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-9H-purin-2-amine
2-[2-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-2-yl)ethyl]pyridine
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
4-cyclopentyl-N-[3-(oxolan-3-yl)propyl]pyrimidin-2-amine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]ethan-1-one
1-[2-methoxy-4-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-phenyl-3-({1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazol-4-yl}formamido)propanamide
4-[3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanoyl]piperazin-2-one
3-ethoxy-N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-4-(prop-2-en-1-yloxy)benzamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(3-methyl-1,2-oxazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-4-phenyl-9-(pyrimidin-2-yl)-2,9-diazaspiro[5.5]undecane
N-[3-(1H-imidazol-1-yl)propyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(ethylamino)pyrimidine-5-carboxamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
[(2S)-1-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-2-yl]methanol
N-(2-methoxyethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-[1-(pyridin-4-yl)propyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-fluorobenzamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(isoquinolin-5-ylmethyl)methylamine
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(propan-2-yl)propanamide
1-({1-[(2-cyanophenyl)methyl]piperidin-3-yl}methyl)-3-(propan-2-yl)urea
7-[2-methyl-2-(thiophen-2-ylformamido)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]pyridine-2-carbonitrile
2-[1-(1-benzofuran-5-carbonyl)piperidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
8-(5-chloro-2-methoxybenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,9R)-11-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
5-(thiophen-3-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
2,5-dimethyl-3-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrazine