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N-methyl-N-[2-(methylamino)ethyl]-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
4-{3-[2-(4-fluorophenyl)azetidin-1-yl]-2,2-dimethylpropyl}morpholine
[3-(1H-1,3-benzodiazol-1-yl)propyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
2-butyl-4-methyl-N-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]-3-oxopiperazine-1-carboxamide
N-methyl-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-[3-(2-methoxybenzamido)phenyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2-(1H-1,2,4-triazol-1-yl)benzamide
4-chloro-1-methyl-3-[1-(pentan-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
2-[1-(2-amino-6-methylpyridin-3-yl)-1H-pyrazol-4-yl]ethan-1-ol
(3R,5S)-N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-3-carboxamide
1-(3-fluorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
N-[(2-methoxyphenyl)methyl]-5-methyl-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]methylamine
5-[4-(adamantan-2-yl)piperazin-1-yl]-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(prop-2-en-1-yl)-5-[4-(propan-2-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-benzyl-N-(1,2-oxazol-3-ylmethyl)-1,3-thiazole-4-carboxamide
4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-1-(2-methoxyethyl)piperidine
7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(pyridin-3-yloxy)phenyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-3-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
N'-(3-chloro-4-methylphenyl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}propanediamide
9-(5-ethyl-1H-pyrrole-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-chloro-2-methoxybenzoyl)-4-(hydroxymethyl)azepan-4-ol
N-(2-methoxy-6-methylphenyl)-4-(2-methoxyphenoxy)piperidine-1-carboxamide
1-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
2-methoxy-N-{2-methyl-3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenyl}acetamide
N-cyclohexyl-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}benzamide
(3S,4R)-4-(hydroxymethyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-ol
(1S,4S)-5-[(2R)-2-amino-3-methoxypropanoyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-{4-[(2-hydroxyethyl)[(2-methylphenyl)methyl]amino]piperidin-1-yl}ethan-1-one
1-cyclopentyl-4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-fluorobenzamide
methyl[(3-methylpyridin-2-yl)methyl]{[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
ethyl 5-{[3-(cyclopentylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
1,1-dioxo-N-(4-phenyl-1,2,3-thiadiazol-5-yl)-1λ6-thiomorpholine-4-carboxamide
3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1-methyl-1H-indole
3-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(methylamino)acetamide
5-[1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-2-(trifluoromethyl)pyridine
(1S,5R)-3-(2-methoxypyridine-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-1-{[1-(2-carboxyethyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[(3-methoxyphenyl)methyl]-5-methyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-methyl-4-[1-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-yl)ethyl]piperazine
N-benzyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(2,2,2-trifluoroethyl)acetamide
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide