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2-{4-methyl-6-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]pyrimidin-2-yl}phenol
6-(cyclobutylamino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-(3-methoxypropyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
ethyl (1R,2S)-2-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}cyclopropane-1-carboxylate
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
2-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}methyl)quinolin-8-ol
(2S)-2-amino-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3,3-dimethylbutan-1-one
2-benzyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1,3-thiazole-4-carboxamide
5-[2-methyl-5-(trifluoromethyl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
N-(2-hydroxy-2-phenylethyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(pyridin-4-ylmethyl)acetamide
(3R,4R)-4-cyclobutyl-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-methylpiperidin-4-ol
4-(2H-1,3-benzodioxol-5-yl)-3-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(ethyl)methylamine
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-(2-methoxyethyl)-6-methyl-4-oxo-N-(pyridin-4-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-sulfamoylbutanamide
1-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(2S,4S)-1-cyclohexyl-N-ethyl-4-[3-(1-methyl-1H-pyrazol-4-yl)propanamido]pyrrolidine-2-carboxamide
2-{[4-(2-methoxyphenyl)-5-(1-methyl-5-oxopyrrolidin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(1-{[4-(difluoromethoxy)phenyl]methyl}azetidin-3-yl)-2-methylpiperidine
N-{2-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
4-{[1-(morpholine-4-sulfonyl)pyrrolidin-3-yl]methyl}benzoic acid
4-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
2-[(4aR,7aS)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
4-{5-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
4-chloro-2-[1-(pyridin-4-yl)-1H-pyrazol-3-yl]phenol
1-benzyl-4-[5-(methoxymethyl)thiophene-2-carbonyl]-1,4-diazepan-6-ol
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl][(8-methoxyquinolin-2-yl)methyl]methylamine
methyl 2-[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]benzoate
1-[(2,5-difluorophenyl)methyl]-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-[1-(1H-indol-5-ylmethyl)piperidin-4-yl]-3-methylbutan-1-ol
2-ethyl-4-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyrimidine
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
4-[2-(dimethylamino)benzoyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-(methoxymethyl)-N-[2-(oxolan-3-yl)ethyl]cyclobutane-1-carboxamide
3-chloro-6-{4-[(2-methoxypyridin-3-yl)methyl]piperazin-1-yl}pyridazine
8-(4-cyclopentylpyrimidin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N,5-dimethyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
4-(2-{[6-(morpholin-4-yl)pyrimidin-4-yl]amino}ethyl)benzene-1-sulfonamide
1-(6-chloropyridazin-3-yl)-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
1-cyclopropyl-N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-6-oxopiperidine-3-carboxamide
ethyl 1-benzyl-5-[(2,6-difluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-chloro-5-(4-hydroxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-dihydropyridin-2-one
1-[1-(8-fluoroquinoline-2-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
3-chloro-4-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)phenol
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1,3-oxazole-4-carboxamide
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-(methoxymethyl)pyrrolidine