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5-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
2-phenyl-4-(4-phenyl-1H-imidazol-5-yl)-1,3-thiazole
1-methyl-3-(2-methylpropyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
1-(1-benzylpiperidin-4-yl)-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
3-(hydroxymethyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-ol
4-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]piperazine-2-carboxylic acid
6-(propan-2-yloxy)-N4-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidine-2,4-diamine
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyrimidine-5-carboxylic acid
4-phenyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,2,3,6-tetrahydropyridine
5-(oxolan-2-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-carboxamide
N-{2-[5-(4-methoxy-2,3-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
methyl[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl][(1-methylpiperidin-2-yl)methyl]amine
1-(4-{1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)propan-2-ol
1-(furan-3-ylmethyl)-4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
N-benzyl({3-[(diethylamino)methyl]phenyl}amino)sulfonamide
N-{[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
(1R,5R)-N,N-dimethyl-6-(2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(6-hydroxy-4-{[(thiophen-2-ylmethyl)carbamoyl]methyl}-1,4-diazepan-1-yl)acetic acid
9-ethyl-4-(5-methoxyfuran-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{3-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}acetamide
6-ethyl-1-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
dimethyl(2-{2-[1-(quinoline-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
6-[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{2-[1-(2,6-difluoro-4-methoxybenzoyl)piperidin-2-yl]ethyl}morpholine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1H-indole-5-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
(3aS,6aS)-2-(cyclobutylmethyl)-5-[2-(6-methylpyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(1H-pyrazol-4-yl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]butanamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidine
2-[3-(1,4-oxazepan-4-ylmethyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
6-[3-(1H-pyrazol-1-yl)benzoyl]-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
(4aR,8aR)-7-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
1-(2-methoxyethyl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
8-(4-aminopyrimidin-2-yl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1H-imidazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)methyl]benzamide
(3R,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[2-(3-methoxyphenyl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
ethyl 4-[(4-{[1-(pyridine-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methylphenol
4-methoxy-N-(2-methoxyethyl)-2-{[1-(pyrimidin-2-yl)piperidin-4-yl]oxy}benzamide
5-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,3-benzothiazol-2-amine
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-(piperidin-3-yl)pyrimidin-4-amine
N-(2-hydroxyethyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
1-(2-{1-[(3-chloro-4-ethoxyphenyl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
(1S,5R)-N-(4-methylphenyl)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}propanamide