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4-(1H-pyrazol-1-yl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidine-4-carboxylic acid
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-hydroxy-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-(2-methylphenyl)pyrrolidine-1-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}furan-3-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]acetamide
1-(1'-{2-[cyclopentyl(methyl)amino]acetyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)-2-methoxyethan-1-one
2-methyl-8-[(2-methyl-1-benzothiophen-3-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
4-{[3-(2-chlorophenoxy)propyl](methyl)amino}pyrimidine-5-carboxylic acid
4-benzyl-1-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-1,4-diazepan-5-one
1-(3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophen-2-yl)ethan-1-one
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
3-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-acetyl-N-[(4-chlorophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(2S,4R)-4-cyclobutaneamido-N-ethyl-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxamide
(butan-2-yl)[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](pyridin-4-ylmethyl)amine
2-(3-chloro-4-hydroxyphenyl)-N-[1-(4-fluorophenyl)piperidin-4-yl]acetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}quinoxaline-6-carboxamide
5-(hydroxymethyl)-2-methyl-4-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)pyridin-3-ol
1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one
(3aS,6aS)-5-(1-benzofuran-2-ylmethyl)-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-(2-ethoxyphenyl)-2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
[(3R,5R)-1-(4,5-dimethylthiophene-2-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
[3-(cyclopropylmethyl)-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-3-yl]methanol
3-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}quinoline
(3R,5S)-N-butyl-1-[(3,4-dimethoxyphenyl)methyl]-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
3-ethyl-8-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(3-propoxypiperidin-1-yl)piperidin-1-yl]-5-(trifluoromethyl)pyridine
1-(dimethylsulfamoyl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
3-(2-fluorophenyl)-1-(3-hydroxyazetidin-1-yl)-3-phenylpropan-1-one
methyl 2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-3-methyl-2-oxopiperazin-1-yl]acetate
5-(2,5-dimethylfuran-3-yl)-1-{3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-3-(oxolan-3-yl)-1H-1,2,4-triazole
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-(hydroxymethyl)cyclopropane-1-carboxamide
N'-(3-chloro-4-methylphenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]propanediamide
4-{pyrazolo[1,5-a]pyridin-7-yl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-hydroxybenzoic acid
N-(2-methoxyethyl)-4-methyl-3-{[(propan-2-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5,6-dimethyl-2-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
2-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
methyl 4-(4-{3-[(2-methoxyethyl)carbamoyl]phenoxy}piperidin-1-yl)pentanoate
dimethyl(2-{2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
{[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}dimethylamine
(butan-2-yl)[(2-chlorophenyl)methyl][(3-methyl-1H-pyrazol-5-yl)methyl]amine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]propanamide
5-ethyl-4-{4-[1-(morpholin-4-yl)ethyl]phenyl}thiophene-2-carboxylic acid
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyrazine
5-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-2-methylpyridine