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[1-({1-[(2E,4E)-5-(4-fluorophenyl)penta-2,4-dien-1-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
{2H-1,3-benzodioxol-5-yl[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}dimethylamine
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[3-(2-methyl-1H-imidazol-1-yl)propyl]amine
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methylpiperidin-3-ol
{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
7-(cyclopropylmethyl)-N-ethyl-6-(2-fluoro-4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-3-propyl-1H-pyrazole-5-carboxamide
3-{2-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-{[1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
4-hydroxy-N-[(2S)-2-hydroxypropyl]-2-phenylpyrimidine-5-carboxamide
1-({4-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)piperidine-4-carboxamide
3-[2-(2-ethyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl){[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-[3-(azepan-1-yl)-2-hydroxypropyl]-3-(3-sulfamoylphenyl)urea
N-(oxan-4-yl)-4-(pyridin-3-yl)pyrimidin-2-amine
2-{2-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-cyclopropyl-3-{1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl}propanamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-(trifluoromethyl)pyrimidin-4-amine
2-(4-chlorophenoxy)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
N-(pyridin-3-yl)-3-[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanamide
1-(4-chlorophenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}cyclobutane-1-carboxamide
1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(1R,2S)-2-phenylcyclopropyl]benzamide
6-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
N'-(3-chloro-4-methylphenyl)-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]propanediamide
8-{3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanoyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-methyl-1-benzofuran-5-yl)-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
1-({2-cyclopropyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-3-methoxy-1,2-dihydropyridin-2-one
3-chloro-6-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-2-carboxylic acid
8-[2-(1H-indazol-1-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-methyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
1-methyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(3-fluorophenyl)methyl]piperidine
2-amino-6-(2,5-dimethylfuran-3-yl)-4-(4-hydroxy-3,5-dimethoxyphenyl)pyridine-3-carbonitrile
N-(3-chloro-4-methoxyphenyl)-3-{1-[(4-acetamidophenyl)methyl]piperidin-3-yl}propanamide
1-[2-(pyridin-2-yl)-4-[(thiolan-3-yl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-fluoro-N-[1-(4-methanesulfonylphenyl)ethyl]quinoline-2-carboxamide
1-ethyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyrrolidin-2-one
N-(3-cyclopentylpropyl)-N-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{4-[(2-hydroxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-(2-methylphenyl)propan-1-one
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide
8-(1,3-benzothiazol-2-yl)-1-(1H-imidazol-2-ylmethyl)-1,8-diazaspiro[4.5]decane
N-ethyl-2-(4-fluorophenoxymethyl)-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]benzonitrile
1-[2-methoxy-4-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
methyl 4-(3-{2-[(3-chloro-4-methoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)-4-oxobutanoate
1-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one