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2-ethyl-7-[4-(2-fluorophenoxy)piperidine-1-carbonyl]-1-(3-methoxypropyl)-1H-1,3-benzodiazol-5-amine
(3R,4S)-4-(5-methylfuran-2-yl)-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}pyrrolidin-3-amine
1-[(3,4-dimethylphenyl)methyl]-4-(5-fluoropyridin-2-yl)piperazin-2-one
2-(4-{5-butyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)pyridine
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methyl-1H-imidazol-2-yl)ethyl]amine
2-amino-4-(6-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-6-(pyridin-2-yl)pyridine-3-carbonitrile
N-(2-chlorophenyl)-4-[2-(thiophen-2-yl)acetyl]morpholine-2-carboxamide
N-(2-methoxyethyl)-N'-(4-methylphenyl)-N-(thiophen-2-ylmethyl)ethanediamide
(3R,9aR)-8-[(4-methylphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-({6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazin-3-yl}amino)ethan-1-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(morpholin-4-yl)propyl]amine
1-benzyl-N-methyl-5-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
N-(oxan-4-yl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]thiophen-3-amine
(3S,5R)-1-[(3,4-dimethoxyphenyl)methyl]-N5-(4-fluorophenyl)-N3,N3-dimethylpiperidine-3,5-dicarboxamide
5-{2-[(3S)-3-acetamidopyrrolidin-1-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
2-[1-(2-methylpropyl)-4-(3,3,5,5-tetramethylcyclohexyl)piperazin-2-yl]ethan-1-ol
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(2-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[1-(furan-2-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
3-(1H-imidazol-2-yl)-N-[2-(2-methylpropanesulfonyl)ethyl]benzamide
phenyl (7S,9aR)-7-ethyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-cyclopentyl-1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-[5-(1-acetylpiperidin-2-yl)-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl]acetic acid
4-[2-(methylamino)pyridine-4-carbonyl]-1-(4-methylphenyl)piperazin-2-one
N-methyl-N-[(5-methylfuran-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]propanamide
1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxylic acid
1-[1-(3-fluoropropyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
N-[(3S,4R)-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]pyridazine-3-carboxamide
2-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-amino-1-[2-(3,4-dichlorophenyl)morpholin-4-yl]propan-1-one
3-[5-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(3S,4R)-1-(2-methoxyethyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-(3,4-difluorophenyl)-4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidine
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[(4-fluorophenyl)methyl]pyrrolidine-2-carboxylate
3-(4-fluorophenyl)-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-pyrazole-5-carboxamide
2-{4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]phenyl}ethan-1-amine
2-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(4-fluorophenoxy)acetamide
5-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
3-ethyl-1-(2-phenylethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-cyclopropyl-1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-[2-(3,5-dimethoxyphenyl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide