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4-(2,4-dioxoimidazolidin-1-yl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
N4-cyclopropyl-6-(4-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}piperazin-1-yl)pyrimidine-2,4-diamine
2-[ethyl(methyl)amino]-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
3-methyl-N-[(3R,5S)-1-(pent-2-yn-1-yl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1,2-oxazole-5-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-2-(2-oxopyrrolidin-1-yl)propanamide
6-chloro-3-fluoro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-cyclohexyl-N-[(2-ethoxypyridin-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-(4-{[3-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
1-(dimethylcarbamoyl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
1-methyl-4-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)-1,4-diazepane
2-(4-methoxyphenyl)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
2-[4-({3-[5-(2-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
3,5-dimethyl-4-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
2-(2-{[methyl(3-methylbutyl)amino]methyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-ethyl-3,5-dimethyl-1H-pyrazole-4-carboxamide
3-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-(furan-2-ylmethyl)piperidine
5-[4-(quinazolin-4-yl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-cyclobutanecarbonylpiperidine-4-carboxamide
(2R,3S,6R)-5-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1-[(2-methoxyphenyl)methyl]pyrrolidin-2-one
5-[(2,6-dioxopiperidin-1-yl)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-[1-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-methyl-N-[2-(4-methylphenoxy)ethyl]acetamide
3-(1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
4-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1-(2-methoxyphenyl)-5-methylpiperazin-2-one
2-[(2S,3R)-2-amino-3-hydroxybutanoyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1'-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-{1-[(4-chlorophenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}-3-methylbutan-1-ol
(1S,5R)-6-(5-propyl-1,2-oxazole-3-carbonyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-(4-{4-[2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}thiophen-2-yl)ethan-1-one
N-[(2-ethoxypyridin-3-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(2-hydroxyethyl)acetamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
4-hydroxy-2-(4-methylphenyl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-5-carboxamide
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-methyl-3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-indole
4-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine
4-({2-[1-(oxane-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(dimethylamino)-N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-4-methylpyrimidine-5-carboxamide
5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-2-(4-methoxyphenyl)pyrimidine
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-[(pyrimidin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
1-(cyclopropylmethyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylic acid
1-(3,4-dimethoxyphenyl)-2-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]ethan-1-ol
5-(4-methyl-1,4-diazepan-1-yl)-2-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
2-hydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}acetamide
2-(1-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine