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(3R,4R)-1-[(3-fluoro-4-methoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-phenyl-3-(3-propoxypiperidine-1-carbonyl)-1,2-dihydropyridin-2-one
4-{2-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
4-(isoquinolin-1-yl)-1-methylpiperazine-2-carboxylic acid
N-[4-(morpholin-4-yl)butan-2-yl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
2-(phenylamino)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrimidine-5-carboxamide
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
5-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3,4-dihydroquinazolin-4-one
N-(furan-2-ylmethyl)-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-propylacetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
4-(3-chloro-4-fluorophenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(propan-2-yl)-5-(2,3,4-trimethoxy-6-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
9-[2-(azepan-1-yl)-2-oxoethyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
1-(3,6-dimethyl-1-benzofuran-2-amido)cyclopentane-1-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(3-methoxyphenyl)propanamide
3-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}methyl)piperidin-3-ol
9-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-(cyclopropylmethyl)-5-[(2-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-(4-{3-[(2-phenylethyl)carbamoyl]phenoxy}piperidin-1-yl)acetic acid
(1S,5R)-3-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(1H-pyrazol-5-yl)piperidine
7-(2-hydroxyethyl)-2-[4-(1,3-oxazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
1-{2-[4-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
2-[(1E)-pent-1-en-1-yl]-6-(piperidine-1-carbonyl)pyrazine
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
2-methyl-5-{4-[3-(piperidin-3-yl)benzoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methylacetamide
4-fluoro-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzene-1-sulfonamide
N-(3-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}phenyl)propanamide
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
2-(1H-imidazol-4-yl)-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethan-1-one
2-(4-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-ol
5-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-(4-{[6-(dimethylamino)pyridin-3-yl]methyl}piperazin-1-yl)-N-ethylacetamide
N-cyclopropyl-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-oxo-N-(oxolan-2-ylmethyl)-1-phenyl-N-(pyridin-4-ylmethyl)-2,5-dihydro-1H-pyrazole-3-carboxamide
4-[4-(1H-imidazol-1-ylmethyl)phenyl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-({4-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-1H-indole
(2R)-1-{1-[(4-methylphenyl)amino]cyclopentanecarbonyl}pyrrolidine-2-carboxamide
N-cyclohexyl-3-{[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}benzamide
1-[(2-{[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}phenyl)methyl]pyrrolidin-2-one
2-(dimethylamino)-4-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrimidine-5-carboxamide
5-(2,6-difluorophenoxymethyl)-N-methyl-N-(pyrimidin-4-ylmethyl)-1,2-oxazole-3-carboxamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[(2,2-dimethyloxan-4-yl)formamido]methyl}benzoate
(1S,5R)-6-methyl-3-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(1H-1,2,4-triazol-5-ylmethyl)acetamide