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N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2,3-dihydro-1,4-benzodioxine-6-carboxamide
2-{5-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-4-(pyridin-4-yl)pyrimidin-2-amine
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]propanamide
3-{4-[(2,4-dimethylphenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}propanoic acid
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-3-(2-methylphenyl)pyrrolidin-3-ol
2-(4-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
6-[4-(dimethylamino)azepan-1-yl]pyridine-3-carbonitrile
2,3-dimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-indole-7-carboxamide
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]pyridine-4-carboxamide
N-cyclopropyl-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(prop-2-en-1-yl)-1-[2-(propan-2-yloxy)acetyl]piperidine-3-carboxylic acid
2-amino-8-[2-(4-chlorophenyl)pyrimidin-5-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
9-[(2-ethoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]methyl}benzonitrile
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-3,4-dimethyl-5-sulfamoylbenzamide
N-[(3R,4S)-1-cyclohexyl-4-cyclopropylpyrrolidin-3-yl]-2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-(3-{[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}phenyl)acetamide
ethyl 1-(2-hydroxyethyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 3-(cyclobutylmethoxy)-5-{[(2-methylpyridin-4-yl)methyl]carbamoyl}benzoate
1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-{4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide
5-(morpholine-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
3-(oxolan-3-yl)-5-(2-propoxyphenyl)-1,2,4-oxadiazole
methyl 4-{[1-(diphenylmethyl)-1H-1,2,3-triazol-4-yl]formamido}butanoate
(1S,5R)-6-(2-chlorobenzenesulfonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[2-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-{4-[4-phenyl-1-(pyridin-2-ylmethyl)-1H-imidazol-5-yl]phenyl}acetamide
4-methoxy-2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
N-ethyl-5-({4-[(4-methylphenyl)sulfanyl]piperidin-1-yl}methyl)pyrimidin-2-amine
3-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)-N-(4-methylphenyl)propanamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(4-methylpentan-2-yl)-1,2-oxazole-3-carboxamide
N-methyl-N-[2-(oxan-4-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
5-[(dimethylamino)methyl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]furan-2-carboxamide
1-(furan-2-ylmethyl)-N-[3-(2-hydroxyphenyl)propyl]piperidine-3-carboxamide
N-(2-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}quinolin-5-yl)acetamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]methyl}piperidin-2-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]piperidine
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
2-({3-[(pyridin-3-yl)amino]propyl}amino)propan-1-ol
4-[4-(2-methylpropyl)piperazin-1-yl]-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
5-ethyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-{1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-4-yl}pyrimidin-2-amine
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[3-(methylsulfanyl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide