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3-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[(3-chloro-4-propoxyphenyl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylacetamide
2-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)-8-fluoroquinolin-4-ol
2-{4-[2-(4-chlorophenoxy)ethyl]piperazin-1-yl}pyrimidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
2-ethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)benzamide
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(2-chloro-3,5-difluorophenyl)-3-methylurea
4-(hydroxymethyl)-1-({2-[(2-methylphenyl)methoxy]phenyl}methyl)azepan-4-ol
N-methyl-N-{2-phenyl-1-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]ethyl}thiophene-3-carboxamide
{[4-ethyl-5-(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
1-[(5-ethylfuran-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
3-{2-[4-(2-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
8-methoxy-N-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)-3,4-dihydro-2H-1-benzopyran-3-amine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-(2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
3-ethyl-5-{[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4,5-dihydro-1,2-oxazole
(3S)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-ol
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]propan-1-one
3-[5-(oxolan-3-yl)-1,2,4-oxadiazol-3-yl]-2-phenoxypyridine
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(cyclopropylmethyl)-9-[(3,5-dimethoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{3-[(2,6-dimethylphenyl)carbamoyl]phenyl}-3-methylfuran-2-carboxamide
N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}pyrimidin-4-amine
4-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)pyridine
5-{[benzyl(methyl)amino]methyl}-N-[(1-methylpiperidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-[(1-acetylpiperidin-4-yl)oxy]-N-(furan-3-ylmethyl)-4-methoxy-N-methylbenzamide
N-{[2-(azepan-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,2-dimethyloxane-4-carboxamide
N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-2-(propan-2-yl)pyrimidine-5-carboxamide
N-[2-methoxy-4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
7-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-4-methyl-2H-chromen-2-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
N-{4-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]phenyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
9-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-5-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
3-{[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}-2,2-dimethylpropan-1-ol
6-amino-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]hexan-1-one
3-{[4-(dimethylamino)oxan-4-yl]methyl}-1-[2-(furan-2-ylmethoxy)phenyl]urea
7-(1,3-benzothiazol-2-yl)-4-(1,3-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(4-methylphenyl)methyl]-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}pyridazine-4-carboxamide
methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]{[5-(oxan-2-yl)furan-2-yl]methyl}amine
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
4-{1-[(2-chlorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-ethyl-3,5-dimethyl-1H-pyrazole
4-[(1R,7S)-3-(2,2-dimethylpropyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
(3aS,6aS)-2-cyclohexyl-5-[(5-methyl-1H-imidazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)urea