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3-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-4-methylbenzene-1-sulfonamide
N-[(3-fluoro-4-methylphenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-hydroxyphenyl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
5-{[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-2-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-(4-methoxy-2-methylphenyl)pyridin-4-amine
(2E)-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-3-(thiophen-2-yl)prop-2-enamide
3-[2-(1-benzylpyrrolidin-3-yl)ethyl]-1-(3-chloro-4-methoxyphenyl)urea
7-(3-chlorophenyl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(cyclopropylmethyl)-4-(5-fluoropyridine-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]benzamide
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]ethan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
6-[4-(hydroxymethyl)piperidin-1-yl]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
2-(dimethylamino)-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2-(3-fluorophenyl)acetamide
N-(5-{[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)carbamoyl]amino}-2-methoxyphenyl)-2-methoxyacetamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-amine
5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-4-phenyl-1H-imidazole
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-acetyl-1H-pyrazole-5-carboxamide
N2,N2-dimethyl-N4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
5-(4-hydroxy-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)-N-(2-methylpropyl)-1-benzofuran-2-carboxamide
5-[(2-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)sulfanyl]-1H-1,2,3-triazole
3-(1H-indazol-5-yl)-1-methyl-1-[1-(pyridin-3-yl)pentyl]urea
(2S,4S)-1-cycloheptyl-N-ethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]pyrrolidine-2-carboxamide
1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
2-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
2-[(2-methylprop-2-en-1-yl)oxy]-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]benzamide
1-(azocan-1-yl)-3-[2-methoxy-5-(morpholin-4-ylmethyl)phenoxy]propan-2-ol
benzyl N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
(3aR,6aR)-2-cyclopentyl-5-[(2-methoxypyrimidin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{1-[5-(piperidin-1-ylmethyl)pyridin-2-yl]-3-propylpiperidin-3-yl}methanol
ethyl 4-[2-(dimethylamino)-6-(4-methylthiophen-2-yl)pyridine-3-amido]piperidine-1-carboxylate
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
4-chlorophenyl (7S,9aR)-7-[(4-chlorophenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
(1R,2R,4R)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]cyclohexan-1-ol
(2R,3R)-N-(furan-2-ylmethyl)-2-hydroxy-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-[1-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridine
2-{1-[(2-ethoxyphenyl)methyl]-4-(pyrazin-2-yl)piperazin-2-yl}ethan-1-ol
N-[(2-chlorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3-methylquinoxalin-2-yl)methyl]-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
[3,3-dimethyl-1-(pyridin-3-yl)butyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1,3-diethyl-5-methyl-6-[2-(pyridin-4-yl)-1H-imidazol-1-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl 3-ethyl-2-(2-methoxypyridin-3-yl)-3H-imidazo[4,5-b]pyridine-6-carboxylate