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4-acetyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
(1R,7S)-3-cycloheptyl-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1H-1,2,3-benzotriazole-5-carboxamide
5-(methoxymethyl)-N-({3-methyl-7-[3-(trifluoromethyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
3-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
ethyl 1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,5R)-6-methyl-3-[4-(2-methylpropyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2,5-dimethylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-3-phenylpropan-1-one
1-[2-({5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethyl]imidazolidin-2-one
1-methyl-4-[2-(2-methyl-1H-indol-3-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 5-(3-methyl-4-oxo-3,4-dihydrophthalazine-1-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2R,6S)-1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylpiperidine
7-chloro-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-methylquinolin-2-amine
(3R,4R)-1-[(3,5-difluorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-4-(morpholin-4-yl)butan-1-one
2-(3-{[2-(1H-imidazol-1-ylmethyl)pyrrolidin-1-yl]methyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
8-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3-methylphenoxy)-1-(oxane-4-carbonyl)piperidine
3-cyclopentaneamido-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(1H-indol-3-yl)-N-(prop-2-en-1-yl)propanamide
2-{3,5-dimethyl-4-[(E)-2-phenylethenyl]-1H-pyrazol-1-yl}-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
2-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)-6-methoxyphenol
1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(3-methoxypiperidine-1-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-indole
4-(2,3-dihydro-1H-inden-2-yl)-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-cyclopentyl-4-[(1-methoxybutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylfuran-2-yl)methyl]acetamide
1-[(3-methoxyphenyl)methyl]-4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]piperazin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-3-phenyl-1H-pyrazole-4-carboxamide
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}pyrimidin-4-amine
N-[2-(benzyloxy)ethyl]-4-ethyl-2-methyl-1,3-thiazole-5-carboxamide
1-(4-{[2-(4-methylphenyl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
6-ethyl-N-(2-methoxyethyl)-2-oxo-N-propyl-1,2-dihydropyridine-4-carboxamide
1-methyl-4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperazine
(2S,4R)-4-amino-N-methyl-1-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]pyrrolidine-2-carboxamide
(3S)-N-tert-butyl-2-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)-N-(2-methoxyphenyl)piperazine-1-carboxamide
2-methyl-4-(3-{4-[(pyridin-2-yl)amino]piperidine-1-carbonyl}phenyl)butan-2-ol
(2S,4R)-N-methyl-4-(4-{2-[(phenylcarbamoyl)amino]propan-2-yl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
(2S)-2-methyl-3-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-ol
N-[(3S)-1-benzylpiperidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(morpholin-4-yl)pyridine-3-carboxamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[3-(6-aminopyridin-2-yl)phenyl]ethan-1-one
4-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-1,4-diazepan-2-one
4-chloro-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N,3-dimethylbenzamide