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3-phenoxy-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
6-acetamido-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyridine-3-carboxamide
4-(4-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)but-3-yn-1-ol
N-(oxolan-2-ylmethyl)-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}piperidine-4-carboxamide
5-(4-methylpiperazin-1-yl)-2-(2-phenoxyethyl)-2,3-dihydropyridazin-3-one
diethyl({2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl})amine
1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
1-ethyl-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2R,3R)-3-{[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-[2-(carbamoylamino)acetyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-(1-cycloheptylpiperidin-3-yl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-methyl-4-oxobutanamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3,3-dimethylbutanoyl)piperidine-2-carboxamide
N-(cyclobutylmethyl)-2-[(2-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
(2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
1-cyclobutanecarbonyl-4-[(2E)-2-methylbut-2-en-1-yl]-1,4-diazepane
3-(1-methyl-1H-pyrazol-5-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]propanamide
1-cyclohexyl-N-[(3-methoxyphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-(2,3-dihydro-1-benzofuran-7-yl)-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
(2S,4S)-4-[2-(carbamoylamino)acetamido]-N-ethyl-1-[(2-fluoro-4-methylphenyl)methyl]pyrrolidine-2-carboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
1-(4-benzylpiperazin-1-yl)-3-[1-(2-phenoxyacetyl)piperidin-3-yl]propan-1-one
5-(cyclopropanesulfonyl)-3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[1-(hydroxymethyl)-9-(1H-imidazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-3-(methylsulfanyl)propan-1-one
N-cyclohexyl-3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-N-methylpropanamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)propanamide
4-methyl-2-propyl-6-[4-(pyrimidin-2-yloxy)piperidin-1-yl]pyrimidine
(2S,4R)-4-amino-1-[4-(diethylamino)benzoyl]-N-methylpyrrolidine-2-carboxamide
5-amino-3-(6-ethoxypyridin-3-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
[(3R,4R)-4-[(dimethylamino)methyl]-1-(propane-1-sulfonyl)pyrrolidin-3-yl]methanol
N-(2-chloropyridin-3-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3-(3-methylphenoxymethyl)piperidine
3-(3-chlorophenyl)-N-methyl-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
4-{4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}thiomorpholine
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
1-(cyclopent-3-en-1-yl)-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
7-methyl-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-1-(2-methoxyphenyl)piperazin-2-one
(1R,5R)-6-(cyclobutylmethyl)-3-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-ethyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
N-methyl-N-(pyrimidin-4-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-(3-hydroxypropanoyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]propanamide