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3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
1-{3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
3-(2,5-dimethylphenyl)-4-[1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
6-methyl-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridin-4-one
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1,4-diazepane-1-carboxamide
N-(1-{1-[2-(2-methoxyphenoxy)acetyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
(1S,5R)-3-benzoyl-6-(1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(6-methylpyridazin-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1,2-dimethyl-4-({3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}sulfonyl)-1H-imidazole
2,6-dimethyl-N-[2-(methylsulfamoyl)ethyl]quinoline-3-carboxamide
methyl[(4-{2-[1-(pyridine-2-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-2-(pyrrolidin-1-yl)benzonitrile
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
(4R)-3-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1,3-thiazolidine-4-carboxamide
2-(5-acetylthiophen-3-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]acetamide
1-(2-methoxyacetyl)-N-[1-(pyrazin-2-yl)propan-2-yl]piperidine-4-carboxamide
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
1-{4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-methoxypropan-1-one
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-{4-[(4-acetyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
2-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]benzonitrile
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
1-ethyl-5-[3-(1H-1,2,4-triazol-3-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl 5-(quinoline-8-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[2-(furan-2-yl)ethyl]-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
N-[2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-3-ol
(3S,5R,9R)-5-hydroxy-11-(thiophene-2-carbonyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-[(3S,4R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-propylpyrrolidin-3-yl]acetamide
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
3-[(3R,4S)-1-[(1-ethyl-1H-indol-6-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-methyl-7-oxo-N-[1-(thian-4-yl)piperidin-4-yl]-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
4-cyclohexanecarbonyl-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(2-methylpropanoyl)-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
9-(3-methylbenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2,3-dihydro-1H-inden-5-yl)-5-(2-methyloxolan-2-yl)-1H-1,2,4-triazole
(3aR,6aR)-2-(3-ethoxypropanoyl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-[4-(3-fluorophenyl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-(2,4-dioxoimidazolidin-1-yl)benzamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,4-diazepan-5-one
N2-methyl-N2-[(4-phenoxyphenyl)methyl]pyrrolidine-1,2-dicarboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3,5-dimethoxybenzamide
N-[3-(methylsulfanyl)phenyl]-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide