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3-methyl-8-(5-propyl-1,3,4-oxadiazol-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,3-dihydro-1H-inden-2-yl)-4-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperazine
(1S,6R)-9-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
methyl 2-{5-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetate
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
7-[(1-methyl-1H-pyrazol-4-yl)methyl]-N4-(thiolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N,N-dimethyl-7-(5-methylpyridine-3-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{4-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazin-1-yl}pyrazine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
N-(2-fluorophenyl)-3-[(1-methanesulfonylpyrrolidin-2-yl)formamido]propanamide
N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[(1S,5R)-3-[(4-cyano-5-methyl-1H-pyrrol-2-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperazine
2-butyl-8-(trimethyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-({3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
2-[benzyl({pyrazolo[1,5-a]pyrimidin-3-ylmethyl})amino]ethan-1-ol
1-[1'-(5-propyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-[2-(3-methoxyphenyl)-1-[1-(oxolane-2-carbonyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
(3S,4S)-4-(morpholin-4-yl)-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidin-3-ol
6-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,3-benzothiazole
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
2-(2-chloro-4-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}phenoxy)acetamide
N-(pyridin-3-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-(4-methanesulfonylphenyl)-2-(propan-2-yl)-1,3-benzoxazole
3-(1H-1,3-benzodiazol-1-yl)-1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]propan-1-one
(4aS,7aR)-1-(2-methylbenzenesulfonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[5-(1H-1,3-benzodiazol-1-yl)-2-methoxyphenyl]methanol
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl})methylamine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-6-ethyl-N,2-dimethylquinoline-4-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(1H-imidazole-2-carbonyl)pyrrolidine-2-carboxamide
N-(2,3-dihydro-1H-inden-5-yl)-3-{[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]amino}-5-(methylsulfamoyl)benzamide
{2-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]pyridin-4-yl}methanol
N-[2-(dimethylamino)ethyl]-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
5-(2-fluorophenoxymethyl)-3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1H-pyrazole
4-benzyl-3-ethyl-1-(2-hydroxy-3-methylbenzoyl)-1,4-diazepan-5-one
1-methyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
5-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-3-phenyl-1H-indole
5-[4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenoxy]-1H-1,2,3,4-tetrazole
(2R)-2-acetamido-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
3,5-dimethyl-2-[3-(morpholin-4-yl)azetidine-1-carbonyl]-1H-indole
N-(2-methoxyethyl)-N,5-dimethyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepane-1-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
4-{[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]methyl}-1-(2-methoxyethyl)pyrrolidin-2-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-cyclohexyl-N3-cyclopropyl-N5-[1-(furan-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-2-one