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2-{4-[(3-chlorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
4-{1-[4-phenyl-5-(1,3-thiazol-2-yl)-1H-imidazol-1-yl]butan-2-yl}morpholine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-hydroxypyridine-3-carboxamide
methyl 3-(furan-2-amido)-6-{[methyl(2-methylpropyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
ethyl 3-benzyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
N,8-dimethyl-2-propyl-N-(pyridin-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}urea
2-(benzyloxy)-1-(4-cyclopentyl-1,4-diazepan-1-yl)ethan-1-one
2-(5-acetylthiophen-3-yl)-N-[1-(4-methanesulfonylphenyl)propyl]acetamide
(2S,4S)-4-(4-butyl-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxylic acid
2,8-dimethyl-N-[(1-methyl-1H-pyrazol-5-yl)methyl]quinoline-4-carboxamide
(1R,5R)-6-(3,4-dimethylbenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(methylsulfanyl)acetamide
N-(2-hydroxyethyl)-1-[1-(1H-indol-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(3-methylphenyl)piperidin-4-yl]-4-sulfamoylbenzamide
5-(4-fluorophenyl)-N-[1-(pyridin-4-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
(1R,5R)-6-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
4-methoxy-6-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-[5-benzyl-4-(2-hydroxyacetyl)-2-oxopiperazin-1-yl]benzonitrile
4-(3-chlorobenzoyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
N-cyclopropyl-3-ethyl-5-hydroxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]adamantane-1-carboxamide
2-(1-ethyl-1H-pyrazol-4-yl)-8-methyl-4-(piperidine-1-carbonyl)quinoline
N-cyclopropyl-5-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2S,4S)-4-amino-N-methyl-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)pyrrolidine-2-carboxamide
2-amino-4-(1-methyl-1H-imidazol-5-yl)-6-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
methyl 4-{4-[3-(3-methylpiperidin-1-yl)propanoyl]piperazin-1-yl}benzoate
3-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
1-(carbamoylmethyl)-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
1-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
4-[5-(2-methyl-1-benzofuran-7-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]-1H-pyrazole
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2,5-dimethoxybenzene-1-sulfonamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
4-(4-methyl-1H-pyrazol-1-yl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine-4-carboxylic acid
1-[(6-ethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-N-ethylpyrrolidine-3-carboxamide
2-(pyridin-2-yl)-7-[2-(1H-pyrrol-1-yl)pentanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(2S,4S)-1-[(3-ethoxyphenyl)methyl]-N-ethyl-4-[(3E)-pent-3-enamido]pyrrolidine-2-carboxamide
7-(1H-pyrazole-3-carbonyl)-N-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]pyridin-3-yl}ethan-1-one
(3S)-3-{[5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]amino}azepan-2-one
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
(1-{2-[3-methyl-4-(morpholin-4-ylmethyl)-1H-pyrazol-1-yl]ethyl}piperidin-3-yl)methanol
6-chloro-3-({[3-(1H-indol-1-yl)propyl]amino}methyl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[(5-methyl-2,1,3-benzothiadiazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
N-[4-({[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)phenyl]acetamide