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{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(2-chlorophenyl)methyl]methylamine
4-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-methyl-1,3-thiazole-5-carboxamide
N-[2-(4-fluorophenyl)ethyl]-2,3-dimethoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}benzamide
6-methyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-2-phenylpyrimidin-4-amine
7-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N3-benzyl-N3,N5-dimethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-cyclopentyl-5-(2-methanesulfonylethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazole
1-amino-N-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)cyclobutane-1-carboxamide
2-(2,3-difluorophenoxymethyl)-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1,3-oxazole-4-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(pyridin-2-yl)acetamide
5-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methyl-5-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine-1-carbonyl)pyrimidin-4-ol
(3S,4S)-4-(piperidin-1-yl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-ol
(4aR,7aS)-1-{2-[methyl(propyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-hydroxyphenyl)-4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
1-(2-methylfuran-3-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
N-[2-(1-{3-[4-(dimethylamino)phenyl]propanoyl}piperidin-2-yl)ethyl]acetamide
2-(2-fluorophenyl)-N-{2-[2-(1H-imidazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}acetamide
N-methyl-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl}-N-(propan-2-yl)acetamide
3-{4-[(5-ethylfuran-2-yl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
7-(cyclopropylmethyl)-2-(5-methyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N1,N1-dimethyl-N3,N3-bis(1,3-oxazol-4-ylmethyl)piperidine-1,3-dicarboxamide
7-(cyclobutylmethyl)-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decane
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(2-oxopiperidin-1-yl)ethyl]benzamide
2-(4-methoxy-3-methylphenyl)-N,N-dimethylpyridine-3-carboxamide
3,3,3-trifluoro-1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(pyridin-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(1-{7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
N-[(3S,4R)-1-(3-hydroxynaphthalene-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-[(2-methoxyphenyl)methyl]-3,4-dihydropteridin-4-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]propan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(isoquinolin-5-ylmethyl)piperidin-3-ol
1-(5-amino-1H-pyrazole-3-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
6-chloro-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
2,3,6-trimethyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]quinoline-4-carboxamide
3-(3-methoxyphenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
4-(piperidin-1-ylmethyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
2-[2-({3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)phenoxy]-N,N-dimethylacetamide
2-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
1-ethyl-N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}piperidine-2-carboxamide
N-(4-hydroxybutyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(2-oxopropanoyl)piperidin-4-yl]oxy}benzamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
2-(2,4-dichlorophenoxy)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
1-{1'-[2-(cyclopent-2-en-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
5-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine