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3-{4-[1-(3-methoxyphenyl)-1H-imidazol-2-yl]phenyl}prop-2-yn-1-ol
(1S,5R)-3-(3-chloro-2-methylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4S)-1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3,3,4-trimethylpiperidin-4-ol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-(1,4-diazepane-1-carbonyl)-N-(2-ethoxyethyl)benzene-1-sulfonamide
methyl (2S)-2-{[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-methylbutanoate
(2R,3R)-3-[4-(pyrazin-2-yl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-(1H-imidazol-4-ylmethyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
N4-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N1,N1,N4-trimethylpiperidine-1,4-dicarboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
(2S,4S)-4-amino-N-methyl-1-(2,3,4-trimethoxybenzoyl)pyrrolidine-2-carboxamide
(3R,4S)-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)-4-phenylpyrrolidin-3-amine
N-methyl-5-{[methyl(oxan-2-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(3-methylfuran-2-carbonyl)piperidin-3-ol
(4aS,8aS)-2-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-7-cyclobutanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
5,7-dimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrido[2,3-d]pyrimidin-4-amine
4-{[2-(difluoromethoxy)phenyl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(3E)-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]hept-3-enoic acid
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(1,3-thiazol-4-yl)acetamide
2-[9-(1-methyl-1H-pyrazole-5-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamide
3-(2-methoxyphenyl)-6-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyridazine
[3-({1-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-4-(thiophen-2-ylmethyl)piperazine
(2S,4R)-4-amino-N,N-diethyl-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxamide
4-(cyclopropylmethyl)-1-[2-(1H-imidazol-2-yl)benzoyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
8-[(5-chlorofuran-2-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(pyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazole
4-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-2-(trifluoromethyl)morpholine
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanoic acid
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
5-(4-chloro-1H-pyrazol-3-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
N-(2H-1,3-benzodioxol-5-yl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
4-(3-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}phenyl)-4H-1,2,4-triazole
N-{4-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]-2-methylphenyl}furan-2-carboxamide
3-methyl-2-{[2-(morpholine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-1H-indole
(3R,9aR)-3-(hydroxymethyl)-8-[(5-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{4-[2-(2-methoxyethyl)morpholine-4-carbonyl]phenyl}-2-methylbutan-2-ol
(4S)-1-(3,5-difluoropyridine-2-carbonyl)-3,3,4-trimethylpiperidin-4-ol
N-(2-ethyl-1H-1,3-benzodiazol-6-yl)-3-(pyridine-2-carbonyl)piperidine-1-carboxamide
N-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
ethyl 2-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamido)acetate
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-ethyl-N-(1-ethylpiperidin-4-yl)-4-methyl-N-[2-(pyridin-2-yl)ethyl]-1,3-oxazole-5-carboxamide