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4-(1-methyl-1H-imidazol-2-yl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
N-[phenyl(pyridin-4-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
N-[1-(2,5-difluorophenyl)cyclopropyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}imidazolidin-2-one
3-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
6-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyridine-3-carboxamide
2-[3-({6-methylimidazo[1,2-a]pyridin-2-yl}formamido)propanamido]acetic acid
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-(3,4-dimethoxyphenyl)piperidin-3-amine
N-[(2-methylphenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)-N-(oxolan-2-ylmethyl)acetamide
2-(4-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}phenoxy)pyrimidine
1-(carbamoylmethyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-4-carboxamide
3-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-(2-phenylethyl)benzamide
1-(5-acetyl-2-ethoxyphenyl)-3-[3-(1H-imidazol-1-yl)propyl]urea
(4aR,7aS)-1-(2-hydroxyethyl)-4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
[(3R,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
{1-[2-(3-methyl-4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-ylmethyl}-1H-pyrazol-1-yl)ethyl]pyrrolidin-3-yl}methanol
2-[(4-hydroxyquinazolin-2-yl)sulfanyl]-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
2-[(1S,5R)-3-(3-acetylbenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}pyrimidin-2-amine
6-(3-hydroxy-4-methoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
2,6-dioxo-N-[2-(3-phenylpropoxy)phenyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
[2-(4-chlorophenyl)ethyl]({[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl})amine
4-(1-ethyl-1H-imidazol-2-yl)-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine
(1S,5R)-6-methyl-3-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
N-(2-hydroxyethyl)-2-[methyl(piperidin-4-yl)amino]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-(pyridin-2-ylmethyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-[(2-chlorophenyl)methyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-(dimethylamino)-4-methyl-N-[2-(1H-pyrrol-1-yl)ethyl]pyrimidine-5-carboxamide
2,4-dimethyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
N-{3-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenyl}propanamide
[(3R,4S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(2S)-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(5-acetylthiophen-3-yl)-1-[2-(2-methylphenyl)pyrrolidin-1-yl]ethan-1-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-phenylpropan-1-one
2-[2-(azocan-1-yl)-2-oxoethyl]-2,3-dihydro-1H-indazol-3-one
ethyl 5-(prop-2-en-1-yl)-1-[3-(pyridin-3-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
3-[(3R,4S)-4-(dimethylamino)-1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]propan-1-ol
3-(2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
5-(3-methylbutyl)-5-(piperidin-4-yl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
1-[(5-chloro-3-methoxy-2-propoxyphenyl)methyl]-4-(hydroxymethyl)azepan-4-ol
N-cyclopropyl-4-methoxy-3-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide