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2-(5-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}furan-2-yl)benzonitrile
2-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-imidazol-2-yl}benzoic acid
N-{[1-(2H-1,3-benzodioxol-5-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-2-methoxyacetamide
2-[(E)-2-cyclohexylethenyl]-5-fluoro-N,N-dimethylpyrimidin-4-amine
(4aS,8aR)-6-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-1-propyl-decahydro-1,6-naphthyridin-2-one
1-methyl-2-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-1H-1,3-benzodiazole
5-(3-methylbut-2-en-1-yl)-1'-(6-methylpyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-3-(5-methylfuran-2-yl)-N-(quinolin-5-ylmethyl)-1H-pyrazole-5-carboxamide
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
6-ethyl-3-(1-hydroxypropan-2-yl)-3,4-dihydroquinazolin-4-one
N-[2-(2-fluorophenyl)ethyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-[(1-benzofuran-2-ylmethyl)(propan-2-yl)amino]propanamide
(benzylsulfamoyl)(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}[(2-phenyl-1,3-oxazol-4-yl)methyl]amine
(4aS,8aS)-2-[(2-butoxy-3-methoxyphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-{2-[(pyridin-3-yl)amino]ethyl}urea
1'-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-(butan-2-yl)-4-oxo-N-(prop-2-en-1-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidine
1-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-(ethylamino)-N-(furan-2-ylmethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
5-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
(4aS,8aR)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
(4S)-4-phenyl-3-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-oxazolidin-2-one
4-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1-methyl-2-phenylpiperazine
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-4-(piperidin-1-yl)butanamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5-methyl-1H-indole-2-carboxamide
4-fluoro-2-methyl-N-[(3R,4S)-1-[2-(methylcarbamoyl)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]benzamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-phenylquinazolin-4-amine
1-cyclohexyl-4-(furan-2-ylmethyl)-1,4-diazepane-6-carboxylic acid
4-methyl-6-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrimidin-2-amine
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
3-[(4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
2-[3-({[1-(2,4-dimethoxyphenyl)ethyl](methyl)carbamoyl}amino)phenyl]-N-methylacetamide
1'-(2,5-dimethylfuran-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)sulfonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-methyl-5-(propan-2-yl)pyrimidine
1-{4-[(2,2-dimethylmorpholin-4-yl)methyl]-2-methoxyphenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
N-(1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
1-methyl-4-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]-1,4-diazepane
N,N-diethyl-1-({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
ethyl 1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
5-{2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-benzoyl-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]piperidin-4-amine
6-methyl-N4-[5-(morpholin-4-yl)pentyl]pyrimidine-2,4-diamine
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl (2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-[(propan-2-yl)carbamoyl]pyrrolidine-2-carboxylate
hexyl(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine