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N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(methylsulfanyl)acetamide
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}oxolane-2-carboxamide
2-oxo-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-2,3-dihydro-1H-imidazole-4-carboxamide
3-(3-fluorophenyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-2-one
7-(1-benzothiophen-3-yl)-4-(1H-pyrazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-[2-(4-chlorophenoxy)ethyl]pyrimidin-4-amine
4-{3-[2-(4-fluorophenyl)azetidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
1-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}piperidine-4-carboxamide
(3S,4S)-4-({[6-(piperidine-1-carbonyl)pyrazin-2-yl]amino}methyl)piperidin-3-ol
1-(2-methyl-4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}phenyl)pyrrolidin-2-one
3-({[1-(oxane-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
6-[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]pyridine-2-carbonitrile
2-[1-(4-fluoro-2-methylbenzoyl)-1,4-diazepan-6-yl]acetic acid
4-[7-(5-propyl-1,2-oxazole-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
4-methyl-1-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydroquinolin-2-one
2-ethyl-8-[3-(1H-imidazol-2-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-({5-[(5-acetylthiophen-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-cyclopropyl-5-{1-[2-(propylsulfanyl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-[2-(3-fluorophenyl)ethyl]-N-(2-hydroxyethyl)-6-oxopiperidine-3-carboxamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
2-butyl-8-{imidazo[1,2-a]pyridine-3-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
N-{[4-(hydroxymethyl)phenyl]methyl}-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
3-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3-methylphenyl)-5-[1-(oxan-4-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
7-methoxy-3-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-1-ethyl-1H-pyrazole-4-carboxamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-[(2-methylphenyl)sulfanyl]acetamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-N-(propan-2-yl)acetamide
2-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]-N-(1,3-thiazol-2-yl)propanamide
3-(2-methoxyphenyl)-N-[2-(4-methylpyrimidin-2-yl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
({4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1,3-thiazol-2-yl}methyl)dimethylamine
N-[4-(3-methyl-1H-1,2,4-triazol-5-yl)phenyl]acetamide
N-(2-chlorophenyl)-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]propanamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-imidazole-5-carboxamide
methyl 2-[2-oxo-4-(quinoxaline-2-carbonyl)piperazin-1-yl]acetate
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-[2-methyl-2-(morpholin-4-yl)propyl]propanamide
2-[3-(4-aminoazepane-1-carbonyl)phenyl]-4-methyl-1,2-dihydrophthalazin-1-one
1-methyl-3-(pyridin-2-yl)-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-1-methylpiperazin-2-one
5-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indazole
7-(4-phenyl-1H-imidazole-5-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[3-(morpholin-4-yl)propyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}acetamide
2-methyl-6-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N-(1-{1-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide