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1-[1-(1H-indol-5-ylmethyl)piperidin-4-yl]-2-phenylethan-1-ol
1-(5-hydroxypentyl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
(2S,4R)-4-{[(2,5-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
2-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]-N,N-dimethylacetamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
3-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
3-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
1-methyl-4-({[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)piperidin-4-ol
2-(4-chlorophenyl)-2-hydroxy-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
N-[(2R,3R)-2-methoxy-1'-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
(1R,3S,5S)-8-{2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carbonyl}-8-azabicyclo[3.2.1]octan-3-ol
2-(1-ethylpiperidin-4-yl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)acetamide
8-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
7-{[(cyclopropylmethyl)(2-methoxyethyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
(3S,7S)-5-(1,3-thiazol-2-yl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(4-methanesulfonylphenyl)-3-(pyrrolidine-1-carbonyl)pyridine
2-(adamantan-1-yl)-N-[2-(1H-imidazol-1-yl)ethyl]acetamide
4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(3-hydroxypropanoyl)piperidin-4-yl]oxy}benzamide
N-(1,3-benzoxazol-2-ylmethyl)-5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(thiophene-3-carbonyl)piperidin-3-amine
2-methyl-5-{4-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
6-[({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amino]pyridine-2-carbonitrile
2-acetamido-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
N-[2-(4-chlorophenyl)ethyl]-2-{methyl[1-(pyrimidin-4-yl)ethyl]amino}acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(2,2,2-trifluoroethyl)benzamide
6-(adamantane-1-carbonyl)-1-(4-benzylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
2-cyclopropyl-4-methyl-5-[4-(pyridin-4-yl)piperazine-1-carbonyl]pyrimidine
[(1R,3S,3aS,6aR)-3-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-(6-phenoxypyridin-3-yl)urea
(1S,6R)-9-{[4-(diethylamino)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylbenzamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-{[1-(5-methylpyridine-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
5-(morpholin-4-ylmethyl)-N-[1-(thiophen-3-yl)propan-2-yl]furan-3-carboxamide
3-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}butanamide
4-(3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-(3,5-dimethylphenyl)piperazin-2-one
N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
N-(5-fluoro-2-methylphenyl)-2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)acetamide
3-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
6-methyl-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-cyclohexyl-4-[2-(oxolan-2-ylmethoxy)acetyl]piperazin-2-one
3-benzyl-8-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(3-methoxyphenyl)sulfanyl]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
(2S,4R)-4-amino-1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
6-methyl-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide