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3-{5-[(2-fluoro-4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-5-methyl-1,2-oxazole
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-(2-chloro-5-methylphenyl)-3-{[1-(hydroxymethyl)cyclopentyl]methyl}-3-methylurea
3-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(3-ethoxyphenyl)urea
4-(5-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidin-2-yl}thiophene-2-carbonyl)piperazin-2-one
1-(1-benzofuran-5-carbonyl)-4-phenyl-1,4-diazepane
3-{5-[(4-methyloxan-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
N-ethyl-N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]naphthalene-2-carboxamide
[(3-chloro-4-methoxyphenyl)methyl](methyl)(oxan-4-ylmethyl)amine
4-[1-(pyrazin-2-yl)propan-2-yl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
N-(1-methyl-1H-pyrazol-4-yl)-2-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}acetamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]acetamide
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-3-(1-methylpiperidin-2-yl)propanamide
ethyl 1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
2-methyl-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}thieno[2,3-d]pyrimidin-4-amine
3-{1-[1-(isoquinolin-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
4-methyl-2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
2-({2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-cyclopropyl-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(methylsulfanyl)propyl]pyrrolidine-3-carboxylic acid
N-[(2,5-dimethylphenyl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-1-(naphthalen-2-ylmethyl)-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
[1-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)piperidin-2-yl]methanamine
{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-3-ylmethyl)amine
N-benzyl-4-(furan-2-carbonyl)piperazine-1-sulfonamide
2-[2-(dimethylamino)ethyl]-9-(5-methylpyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)phenyl]formamido}ethyl)piperidine-3-carboxamide
2-(1,3-benzoxazol-2-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(3aR,6aS)-2-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole
2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}quinoxaline
1-phenyl-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-2-one
4-methyl-1-(2-phenylpropyl)-1,4-diazepan-5-one
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-1H-indazole-3-carboxamide
2-benzyl-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(2,3-difluorophenyl)methyl]-2-(prop-2-ene-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[3-(4-fluorophenyl)benzoyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-[(prop-2-en-1-yl)amino]-N-(pyridin-4-ylmethyl)benzamide
N-benzyl-N,1-dimethyl-5-{[3-(methylsulfanyl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-5-(3-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
2-{2-[4-(3-fluorophenoxy)piperidin-1-yl]ethyl}-2H-indazole
1-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-1,2,3,4-tetrahydroquinolin-2-one
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S)-2-amino-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-phenylethan-1-one
1-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}imidazolidin-2-one
N-methyl-N-phenyl-2-(4H-1,2,4-triazol-4-yl)benzamide
2-{[2-(2-hydroxyethyl)morpholin-4-yl]methyl}-6,8-dimethylquinolin-4-ol
1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-({1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}methyl)acetamide
N-methyl-N-[4-(morpholin-4-yl)butyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-[(dimethylamino)methyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]azepan-4-ol