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4-(benzyloxy)-1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butan-1-one
N-({1-[(4-methylphenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)acetamide
1-(diethylamino)-3-(2-methoxy-5-{[methyl(3-methylbutyl)amino]methyl}phenoxy)propan-2-ol
[(3R,4S)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(2R,4R,6S)-2-(4-chlorophenyl)-6-{pyrazolo[1,5-a]pyrimidin-3-yl}oxan-4-yl]acetamide
2-cyclopropyl-8-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-1-methylurea
N-methyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-4-(trifluoromethoxy)benzene-1-sulfonamide
(4aR,8aR)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridine
2-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}-N-[1-(4-methylphenyl)ethyl]acetamide
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-N-methylpyridin-2-amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-2-one
(2S,4R)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-(2-phenylacetamido)pyrrolidine-2-carboxamide
2-oxo-N-(propan-2-yl)-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)acetamide
2-{3-[(2,6-dichlorophenyl)methyl]-5-(pyrrolidin-3-yl)-1H-1,2,4-triazol-1-yl}acetic acid
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
ethyl 1-benzyl-5-(1H-indol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-benzyl-4-(6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-sulfonamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(1-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)-1H-1,3-benzodiazole
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S)-2-cyclohexyl-2-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]acetic acid
(2S,4R)-1-[(4-chlorophenyl)methyl]-N-(propan-2-yl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-benzyl-2-(dimethylamino)-4-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrimidine-5-carboxamide
1-[(4-methylphenyl)methyl]-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazin-2-one
2-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(1-phenoxyethyl)-5-{pyrazolo[1,5-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(furan-2-yl)-7-methyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-hydroxy-1-(thian-4-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(1-methylpiperidine-2-carbonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylic acid
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-(quinolin-2-ylmethyl)propanamide
2-[2-benzyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]acetamide
ethyl 1-[3-(2,5-dioxoimidazolidin-4-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
4-(4-chlorophenoxy)-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]piperidine-4-carboxamide
N2-ethyl-N2-{[3-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-1,2-dicarboxamide
2-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]pyridine-4-carboxamide
9-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(methylsulfanyl)phenyl]methyl}-N-propyl-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-(propan-2-yl)pyridazine
8-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-phenyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(3aR,6aR)-2-(2-aminopyrimidin-4-yl)-5-(3-methylbut-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N1,N1-dimethyl-N3-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-1,3-dicarboxamide
1-{2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}azepan-2-one
2-(2-cyclopropylacetyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-methyl-N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
2-[4-(4-carbamoylpyridin-2-yl)phenoxy]acetic acid