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2-benzyl-9-[(1R,2S)-2-propylcyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
6-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]acetamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
(3aR,6aR)-2-cyclopentyl-5-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(1H-pyrazol-4-yl)benzamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(piperidin-4-ylmethyl)benzamide
3-(2-methoxyphenyl)-N-[2-(1-methylazepane-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
2-(2-methoxyethyl)-8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-butyl-4-(2-fluoro-6-methoxybenzoyl)-1-methylpiperazin-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]piperidin-2-one
N-(6-chloropyridin-3-yl)-4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carboxamide
6-methyl-5-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-phenoxypropan-1-one
N-{2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}-2-methylpropanamide
methyl 1-{2-hydroxy-3-[4-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]pyridin-3-ol
8-(3-chloropyridin-2-yl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(2-phenyl-1,3-thiazol-4-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-(furan-3-ylmethyl)urea
N-(4-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}-3-methylphenyl)acetamide
2-cyclopentyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(propane-1-sulfonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[5-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]acetic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-methylpiperidine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(dimethoxy-1,3,5-triazin-2-yl)thiophene-2-carboxylic acid
(4-{[4-(3-cyclohexyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
(4aS,7aR)-1-(5-ethylthiophene-3-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(5-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethylpyrimidine-5-carboxamide
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-(4-methylphenoxymethyl)piperidine
1'-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-[3-(5-chlorothiophen-2-yl)phenyl]-4H-1,2,4-triazole
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(3,4-difluorophenyl)methyl]piperazin-2-one
4-(4-chlorophenoxy)-1-(6-cyanopyridin-2-yl)piperidine-4-carboxylic acid
3-[3-(2-phenylethyl)piperidine-1-carbonyl]pyridine
1-cyclopentanecarbonyl-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
N-(3-chloro-4-fluorophenyl)-3-(1-cyclopentanecarbonylpiperidin-4-yl)propanamide
ethyl 1-{[4-(methoxycarbonyl)phenyl]methyl}-4-(2-methoxyethyl)piperidine-4-carboxylate
4-(3-hydroxypropyl)-11-{[(1-phenylcyclopentyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[2-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)ethyl]piperidine-3-carboxamide
3-[5-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]acetyl}-1-phenylpiperazin-2-one
6-chloro-2-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]quinolin-4-ol
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(1-hydroxypropan-2-yl)acetamide
3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
2-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido