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1-[4-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amino}methyl)thiophen-2-yl]ethan-1-one
(3R,4R)-7-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-3-(pyrrolidin-1-yl)-3,4-dihydro-2H-1-benzopyran-4-ol
3-(azocan-1-yl)-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)propanamide
N-[2-(1H-pyrazol-1-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(4-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-[2-(3,4-difluorophenyl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
1-[(4-methanesulfonylphenyl)methyl]-3-phenylpiperidine
7-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}-2-oxa-7-azaspiro[4.5]decane
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
N-(1-hydroxy-2-methylpropan-2-yl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[3-(1,3-benzothiazol-2-yl)propyl]-5-ethyl-1,3,4-oxadiazol-2-amine
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-methyl-2-(4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
4-[(1E)-3-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}prop-1-en-1-yl]-2-methoxyphenol
methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl][2-(pyridin-2-yl)ethyl]amine
(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-N-phenyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(3aS,6aS)-2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5-[2-(pyridin-4-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(4-methoxyphenoxy)piperidine
(2S,4R)-4-[4-({[(2,5-difluorophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-(4-{[(1R,5S)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(oxan-3-ylmethyl)acetamide
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N,N-dimethylpiperazine-1-sulfonamide
14-(4-methoxy-2,5-dimethylphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-(1H-imidazol-1-yl)-N-({3-methyl-7-[(2E)-3-phenylprop-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)acetamide
11-(1H-indol-2-ylmethyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-5-fluoro-1H-1,3-benzodiazole
8-[5-(cyclopentylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]quinoline
N-ethyl-5-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)pyrimidin-2-amine
1-(3-chlorophenyl)-4-(1,4-dioxane-2-carbonyl)piperazine
1-[(3-chloro-4,5-diethoxyphenyl)methyl]piperidine-4-carboxamide
5,6-dimethoxy-2-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-1,2-dihydroisoquinolin-1-one
2,5-dimethyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
N-ethyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[5-(oxan-2-yl)furan-2-yl]methyl}amine
({5-[(adamantan-1-ylsulfanyl)methyl]-1,2,4-oxadiazol-3-yl}methyl)dimethylamine
1-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]azetidin-3-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(2-methyl-1H-imidazol-1-yl)propanamide
1-(2-methoxyphenyl)-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}-1λ6-thiomorpholine-1,1-dione
N-[(1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)methyl]acetamide
4-{2-[3-(2,6-dimethylphenoxy)azetidin-1-yl]pyridine-4-carbonyl}morpholine
2-(2-aminoethyl)-5,6-dimethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)thieno[2,3-d]pyrimidin-4-amine
(3aS,6aS)-2-(cyclopropylmethyl)-5-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(oxan-4-yl)pyridin-2-amine
5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]pyrazin-2-ol
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-N,N-dimethylaniline
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)piperidin-2-one
4-(4-fluorophenyl)-N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,6-tetrahydropyridine-1-carboxamide