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1-[3-(2-{[(2,2-dimethylpropyl)(methyl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-3-yl]propanoate
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(3,4-difluorophenyl)methyl]piperidine
5-(5,6-dimethylpyrazin-2-yl)-2-methylquinoline
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{5-[(2S)-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
6-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(3-fluorophenyl)methyl]urea
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-(1H-pyrazol-1-yl)butanamide
1-(2-ethylpyridine-4-carbonyl)-4-[(2-methylphenyl)methyl]piperazine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1S,2R)-2-aminocyclobutyl]acetamide
(3S,4R)-4-methyl-1-(5-propylpyrimidin-4-yl)piperidine-3,4-diol
6-(benzyloxy)-1-cyclohexyl-4-cyclopropanecarbonyl-1,4-diazepan-2-one
N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)benzamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,5-dimethyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-[(2,6-dimethoxyphenyl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 3-[(3-hydroxy-4-methoxyphenyl)methyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]ethan-1-one
3-(2-methylphenyl)-3-phenyl-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
7-cyclobutanecarbonyl-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-6-methylpyridine-3-carboxamide
ethyl 1-[3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanoyl]piperidine-2-carboxylate
2-(2-aminoethyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]quinazolin-4-amine
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(2,2,2-trifluoroethyl)piperazine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
1-[2-(3,4-dimethylphenoxy)ethyl]-4-(1-ethyl-1H-imidazol-2-yl)piperidine
1-(1-acetylpiperidin-4-yl)-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
7-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}({[5-(methoxymethyl)furan-2-yl]methyl})amine
N-ethyl-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-methoxyethyl)-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-[cyclopentyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]acetic acid
4-(4-chlorophenoxy)-1-(oxan-4-yl)piperidine-4-carboxylic acid
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](furan-2-ylmethyl)methylamine
3-[1-(quinoxalin-5-ylmethyl)piperidin-3-yl]propanamide
3-(4-hydroxyphenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[2-(furan-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[1-(4-methanesulfonylphenyl)propyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
3-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
ethyl 1-(benzylsulfamoyl)piperidine-4-carboxylate
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
4-[2-(3-chlorophenyl)ethyl]-11-(cyclopentylamino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl (2S)-1-{2-[4-(4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
3-[6-(dimethylamino)pyrimidin-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
1-(azepan-1-yl)-3-[(6-methoxypyrimidin-4-yl)amino]propan-2-ol
N-methyl-3-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}propanamide