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N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(3-carbamoylpiperidin-1-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-ethoxy-3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine
(1R,6S)-9-methyl-3-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3,9-diazabicyclo[4.2.1]nonane
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3,3,3-trifluoropropyl)acetamide
3-(4-{4-[(tert-butylcarbamoyl)amino]phenyl}-3,5-dimethyl-1H-pyrazol-1-yl)propanamide
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-4-(trifluoromethyl)pyrimidin-2-amine
methyl (1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
N-[3-(1H-indazol-1-yl)propyl]-2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
3-(2-hydroxyphenyl)-N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
2-(1-butyl-1H-pyrazol-4-yl)-N,N,3,6-tetramethylquinoline-4-carboxamide
4-benzyl-3-ethyl-1-(3-methoxypropyl)-1,4-diazepan-5-one
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3H,4H-pyrido[3,4-d]pyrimidin-4-one
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
6-methoxy-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexan-1-one
5-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(2-methylpropyl)-1-benzofuran-2-carboxamide
6-(2-fluorophenyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
5-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
13-[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
4-hydroxy-1-methyl-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}piperidine-4-carboxamide
1-(6-{4-[(2,6-difluoro-4-methoxyphenyl)methyl]piperazin-1-yl}pyridin-3-yl)ethan-1-one
2-(4-{3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidin-2-yl)phenol
{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-phenylethyl)piperidin-4-yl}methanol
1,3-dimethyl-8-[2-(thiophen-3-yl)acetyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1-{2-[(cyclopropylmethyl)sulfanyl]acetyl}piperidin-3-yl)benzoic acid
[3-(3-methoxypropyl)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]methanol
(3S,4S)-4-(morpholin-4-yl)-1-(3-phenylpropyl)pyrrolidin-3-ol
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-(pyridin-2-ylsulfanyl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethan-1-one
9-(cyclopropylmethyl)-4-[2-(3-fluorophenyl)ethyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4S,5R)-4-[(2-hydroxyethyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
6-[(3-methylpiperidin-3-yl)methoxy]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
7-[4-(3-chlorophenoxy)piperidine-1-carbonyl]-1,3-diazepane-2,4-dione
ethyl 3-[(3-methoxyphenyl)methyl]-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine-3-carboxylate
2-[({5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(1S,6R)-9-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
2-methoxy-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
N-[2-phenyl-2-(piperidin-1-yl)ethyl]thiophene-3-carboxamide
4-{4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
5-(4-fluorophenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2,4-difluoro-3-methoxy-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
(2R,3R)-3-amino-1'-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]pyridine-3-carboxylic acid
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methylpent-3-en-1-yl)piperidine
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]pyridine-4-carboxamide
N-benzyl-2-(4-{4-[methyl(thiophen-3-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
1-(2-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-4-methylpyrimidin-5-yl)ethan-1-one
N-cyclopropyl-1-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]piperidine-2-carboxamide