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1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
3-(1H-imidazol-4-ylmethyl)-4-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperazin-2-one
1-(1-{[3-(benzyloxy)phenyl]methyl}pyrrolidin-3-yl)-4-methylpiperazine
N-cyclopropyl-1-{1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
2-(4-{[(1R,3R)-3-aminocyclopentyl]amino}-6-methylpyrimidin-2-yl)phenol
2-{[ethyl(oxolan-2-ylmethyl)amino]methyl}-6-methoxyphenol
2-(1,4-dimethylpiperazin-2-yl)-N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
(4-{[1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-(5-chloro-2-methoxyphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
3-(3-fluorophenyl)-1-(3-methylphenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
N-[(3R,4S)-1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
2-[5-(5-acetylthiophen-3-yl)-4-phenyl-1H-imidazol-1-yl]-N,N-dimethylethane-1-sulfonamide
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
3-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-benzyl-1H-pyrazole-4-carboxamide
2-benzyl-8-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-methylpropyl)acetamide
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}isoquinoline
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanoic acid
1-[4-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(2-hydroxyethyl)piperidine-4-carboxylate
4-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)thiomorpholine
N-(butan-2-yl)-N-(pyridin-4-ylmethyl)-6-[2-(pyrrolidin-1-yl)ethyl]pyridine-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(thiolan-3-yl)benzamide
1-[4-(4-fluorophenyl)benzoyl]-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
N-[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]acetamide
1-[(3S,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-(benzyloxy)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
5-(methoxymethyl)-N-(3-methylbutyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
methyl 2-(ethylsulfamoyl)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyridine
3-(5-methylfuran-2-yl)-5-[2-(oxolan-2-yl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
(1R,5R)-N-(2H-1,3-benzodioxol-5-yl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine
2-benzyl-8-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
8-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
7-(2-hydroxyethyl)-2-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)ethyl]-N-methyl-3-[(oxolan-3-yl)sulfamoyl]benzamide
3-[1-(1H-imidazol-1-yl)butan-2-yl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
5-chloro-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-phenyl-1H-indole-2-carboxamide
3,6-dimethyl-4-(piperidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
N-ethyl-4-hydroxy-N-[2-(phenylsulfanyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(3,5-dimethylphenyl)-2-{8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-oxoacetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(2-hydroxyethyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
N-(1-phenyl-1H-pyrazol-5-yl)-2-[4-(pyrimidin-5-yl)-1H-pyrazol-1-yl]acetamide
4-[(dimethylamino)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}azepan-4-ol