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(4aS,7aR)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[5-(1,1-dioxo-1λ6-thian-4-yl)-1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
(4aR,7aS)-1-(pyridine-2-carbonyl)-4-(thiophen-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-chloro-2-{[4-(3-methyl-1,2-oxazol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
N-(1-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)pyrimidin-2-amine
1-[(5-chloro-2-hydroxyphenyl)methyl]-4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}piperidin-4-ol
2-{4-cyclobutyl-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methoxypyridine-3-carbonitrile
4-(dimethylamino)-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
(3aS,6aS)-2-cyclopropanecarbonyl-5-[ethyl(methyl)sulfamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-(pyrimidin-4-yl)piperidine-1-carboxamide
4-[(3-methoxypropyl)amino]-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-ethyl-4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
2-(benzyloxy)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
3-benzyl-1-(8-methoxyquinolin-2-yl)piperidine-3-carboxylic acid
N-(3-cyanothiophen-2-yl)-4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)benzamide
3-(2,5-dimethoxyphenyl)-1-ethyl-1-(oxan-4-ylmethyl)urea
(1R,3S)-7-(4,5-dimethylthiophene-2-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
8-{2-[(2-methylphenyl)sulfanyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
2-(2,3-dimethylphenoxy)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
3-[(3,4-dimethoxyphenyl)methyl]-1-ethyl-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-1,2,4-triazole
6-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)-1,4-oxazepan-6-ol
4-({2-[5-(1,4-oxazepane-4-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}methyl)pyridin-2-ol
6-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-2-carbonitrile
6-ethyl-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(morpholin-4-yl)pyrimidin-4-amine
4-[5-({[(2R)-oxolan-2-ylmethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
3-(azocan-1-yl)-N-[3-(1H-imidazol-1-yl)propyl]propanamide
1-(2-{[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
methyl[3-(phenylsulfanyl)propyl]{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(benzyloxy)ethan-1-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-(naphthalen-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-cyclopentanecarbonylpiperidine-4-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-propylacetamide
4-(2-ethoxypyridin-3-yl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
N-methyl-4-(pyrrolidine-1-carbonyl)-6-{spiro[2.3]hexane-1-carbonyl}-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-cyclopropyl-N-({4-methoxy-3-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-4-(trifluoromethyl)benzamide
[(4-methanesulfonylphenyl)methyl](methyl)(1H-pyrazol-3-ylmethyl)amine
5-({[(3-{2-[4-(2-methoxyacetyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
methyl 4-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
2-amino-4-[4-methoxy-3-(methoxymethyl)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
4-[5-(quinolin-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]benzonitrile
6-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-2-propoxypropan-1-one
5-propyl-N-[(1r,4r)-4-hydroxycyclohexyl]-1,2-oxazole-3-carboxamide
(4aS,7aR)-1-[(6-methylpyridin-2-yl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({3-[(dimethylamino)methyl]phenyl}methyl)-N,2,5,6-tetramethylpyrimidin-4-amine