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N-[(2-ethoxypyridin-3-yl)methyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
methyl (2S)-2-({1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-3-(1H-imidazol-4-yl)propanoate
6-methoxy-3-{[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-4-methoxybenzamide
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-3-methyl-1,2-oxazole-5-carboxamide
(4aS,8aR)-6-[2-(benzenesulfonyl)ethyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(1R,3S)-7-[4-(difluoromethoxy)benzoyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-methyl-N-(oxan-2-ylmethyl)-3-(piperidin-4-ylmethyl)benzamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
3-amino-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,4-triazole-5-carboxamide
4-{[4-(4-hydroxyphenyl)butan-2-yl]amino}-N-phenylpiperidine-1-carboxamide
2-(1-{1-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
3-chloro-6-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-(3-methylphenyl)piperidine-1-carboxamide
1-benzyl-3-(oxan-4-yl)-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazole
methyl({1-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
3-({[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}amino)propan-1-ol
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-4H-thieno[3,2-b]pyrrole-5-carboxamide
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
3-{[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
5-methoxy-1-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-indole-2-carboxamide
N-{2-methoxy-5-[({2-[(3-methylpyridin-2-yl)amino]ethyl}carbamoyl)amino]phenyl}propanamide
(1R,2R,6S,7S)-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-[1-(1H-pyrazol-3-ylmethyl)piperidin-2-yl]pyridine
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(3-methoxyphenyl)-3-methylpiperazin-2-one
(3S,4R)-4-(4-fluorophenyl)-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]pyrrolidine-3-carboxylic acid
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
1-[4-(furan-2-yl)phenyl]-N-[2-(1H-imidazol-4-yl)ethyl]piperidin-4-amine
N2,6-dimethyl-N4-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyrimidine-2,4-diamine
2-ethyl-8-(4-methylnaphthalene-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-propyl-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-5-carboxamide
5-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(6-chloropyridin-3-yl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
1-[(3-ethoxyphenyl)methyl]-1-(2-hydroxyethyl)-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
N-(pyridin-2-ylmethyl)-4-(quinolin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[2-amino-4-(cyclopentylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1H-pyrrol-1-yl)ethan-1-one
3-(2-fluorophenyl)-N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-{[5-fluoro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-2-yl)acetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
3-phenyl-1-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
2-(4-fluorophenyl)-1-{9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
1-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-5,5-diphenylpiperidin-2-one
N-(1,4-dioxan-2-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-[2-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-(1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-methyl-1'-(5-methylpyridine-3-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-{[5-(3-fluoropyridin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
3-(azepane-1-carbonyl)-N-[(3-methoxyphenyl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine