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1-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}urea
5-ethyl-2-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyridine
4-{4-[(2,4-dimethoxyphenyl)methyl]piperazin-1-yl}-2-[(1-hydroxycyclohexyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
[(5-{[3-(4-fluorophenoxy)azetidin-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinoxalin-6-ylmethyl)amine
methyl 3-{[(2-fluorophenyl)formamido]methyl}-5-(quinoline-8-sulfonamido)benzoate
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(oxan-3-yl)pyrimidin-2-amine
5,6-dimethyl-3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
6-methyl-2-({[2-(oxan-2-yl)ethyl]amino}methyl)quinolin-4-ol
phenyl (7S,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-[(4,6-dimethylpyridin-2-yl)methyl]-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
3-{5-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
6-(2-ethoxypyridin-3-yl)-N2,N2-diethylpyrimidine-2,4-diamine
2-[1-(2H-1,3-benzodioxol-5-yl)-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-7H-pyrrolo[2,3-d]pyrimidine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyrrolidine-3-carboxamide
8-[(3-chloro-5-fluorophenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
3-benzyl-1-(3-methoxypropyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[2-(1-methylpyrrolidin-3-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-2-carbonitrile
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{thieno[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-({1-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}(methyl)amino)ethan-1-ol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(4,4,4-trifluorobutyl)piperidine
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-[(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
6,9-dioxo-N-(2-phenoxyphenyl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-[1-(4-methanesulfonylphenyl)ethyl]-2-methyl-1-benzofuran-7-carboxamide
N-(2-{1-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]piperidin-2-yl}ethyl)acetamide
2-(5-acetylthiophen-3-yl)-N-[(4-methoxyphenyl)methyl]-N-propylacetamide
2-[4-(7-chloro-2-methylquinoline-4-amido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
6-[4-(1H-pyrazol-5-yl)phenyl]-9H-purine
1-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]-2-phenylethan-1-ol
1-[(2-chlorophenyl)methyl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-benzyl-4-(2-{[(1-ethylpyrrolidin-2-yl)methyl]carbamoyl}ethyl)piperidine-1-carboxamide
1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(4aR,7aS)-1-(cyclopropylmethyl)-4-(2-hydroxy-3-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(5-aminopyridin-3-yl)-3,5-dimethyl-1H-pyrazol-4-yl]propan-2-one
1-[(3,4-difluorophenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(cyclohexylmethyl)-4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
(3S,4R)-1-[4-(morpholin-4-yl)benzoyl]-4-phenylpyrrolidine-3-carboxylic acid
[2-(1H-imidazol-4-yl)ethyl]({[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl})amine
1-{2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[(2,3,4-trimethoxyphenyl)methyl]pyrrolidine-2-carboxamide
5-[4-(3,4,5-trimethoxyphenyl)phenyl]-1H-1,2,3,4-tetrazole
5-{1-[(4-ethylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
1-methyl-N-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[({2-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]methyl}cyclohexan-1-ol
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
5-(1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
8-benzyl-N,N-dimethyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-sulfonamide