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1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)(methyl)amino]methyl}piperidin-2-one
N-(1-benzylpyrrolidin-3-yl)-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-butyl-1-methyl-4-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperazin-2-one
(2S)-3-(1H-indol-3-yl)-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]propanoic acid
N-ethyl-N-(propan-2-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
2-oxo-8-[(2-phenylethyl)carbamoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-methoxy-2-methylpropan-1-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-N'-cyclopentylbutanediamide
(4aR,7aS)-1-pentanoyl-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-5-[3-methyl-1-(2-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-imidazole
2-[(1r,4r)-4-hydroxycyclohexyl]-9-[2-(thiophen-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{4-[6-amino-5-cyano-4-(pyridin-3-yl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}propanoic acid
(2R)-1-({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)pyrrolidine-2-carboxamide
5,5-diphenyl-1-[1-(pyrimidin-4-yl)ethyl]piperidin-2-one
7-[(3,4-difluorophenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decane
2-(2-{1-[4-(dimethylamino)butanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-{4-[2-(phenylsulfanyl)acetyl]morpholin-3-yl}acetic acid
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(1H-pyrazol-1-yl)benzamide
N-(4-fluorophenyl)-1-(thian-4-yl)piperidin-3-amine
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
2-benzyl-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(4-ethoxy-3-methylphenyl)-4-oxobutanamide
methyl[(3-{2-[4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](1,3-thiazol-4-ylmethyl)amine
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
7-methyl-4-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-2H-chromen-2-one
N,3,5,7-tetramethyl-N-[3-(oxolan-2-yl)propyl]-1H-indole-2-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine-4-carboxylic acid
5-{[4-(morpholine-4-carbonyl)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
2-(adamantan-1-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]acetamide
5-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(5-hydroxyadamantan-2-yl)propanamide
1-benzyl-4-(3,3,4,4-tetrafluorobutyl)-1,4-diazepan-6-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
(2R,3S,6R)-3-(4-methylphenyl)-5-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
2-[ethyl({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
1-(2-methylpentyl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-hydroxypropan-1-one
4-{[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenol
N-methyl-7-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-{[7-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
2-amino-6-(1-phenyl-1H-pyrazol-4-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
1-{[3-(propan-2-yl)-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
2-ethyl-8-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}-N,N-dimethylethane-1-sulfonamide
6-[(3S)-3-ethylmorpholine-4-carbonyl]-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one