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N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-(1-benzofuran-2-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-(3-aminopropyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H-1,2,3-triazole-4-carboxamide
8-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
4-({[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}amino)pyrimidine-5-carboxylic acid
3-[(4-fluorophenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
2-(4-methyl-1H-imidazol-5-yl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)-1H-imidazole
(3R,4R)-4-(morpholin-4-yl)-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-ol
N-methyl-N,2-bis(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
2-cyclopropyl-9-(2,3-difluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(1,3-dimethyl-1H-pyrazol-4-yl)-3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-[(3R,4S)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]-N-methylpyridine-3-carboxamide
(2S,4R)-N,N-diethyl-4-[2-methyl-5-(propan-2-yl)furan-3-amido]-1-propylpyrrolidine-2-carboxamide
2-[(1S,5R)-6-(2-chloro-4-fluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-[(5-chloro-2-propoxyphenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-(1H-1,3-benzodiazol-2-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
(1S,5R)-3-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{9-[(5-cyano-1-methyl-1H-pyrrol-3-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
1-(4-methylphenyl)-4-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)pyrrolidin-2-one
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(morpholin-3-yl)acetamide
3-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-1-(furan-2-ylmethyl)piperidine
5-methoxy-1-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-indole-2-carboxamide
N4-{[1-(dimethylamino)cyclohexyl]methyl}-5-methylpyrimidine-2,4-diamine
2-[3-(1H-pyrazol-3-yl)phenyl]-4-(trifluoromethyl)pyrimidine
(2S,4R)-4-(dimethylamino)-1-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidine-2-carboxylic acid
[(3aS,6aS)-2-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]benzene-1,3-diol
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-fluorophenoxy)piperidine
(2S,4R)-1-benzyl-N-ethyl-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
5-(2,2-dimethylcyclopropanecarbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
(2S,4S)-4-amino-1-[(4-acetamidophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
(1S,5R)-6-(3-propyl-1H-pyrazole-4-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(4aR,8aR)-6-[2-(2-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-2-(4-chloro-2-methylphenoxy)ethan-1-one
1-[(2,3-dichloro-4-methylphenyl)methyl]piperidine-4-carbonitrile
4-[3-(methylsulfanyl)butyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3aR,6aR)-2-cyclopropanecarbonyl-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-1-methylazepane-2-carboxamide
2-(2-ethylbutanoyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(4aS,8aR)-6-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
(4aS,8aR)-6-[(2-methylpyrimidin-5-yl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]pyridine-2-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
4-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-[({[5-(hydroxymethyl)furan-2-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2'-oxo-1',2',3',5'-tetrahydrospiro[cyclobutane-1,4'-pyrido[3,2-b]indole]-3-carboxylic acid
4-[2-amino-3-cyano-5-methyl-6-(5-methylthiophen-2-yl)pyridin-4-yl]benzamide
N-benzyl-3-(1-methanesulfonylpiperidin-4-yl)-N-methylpropanamide
N-[(5-chloro-2-propoxyphenyl)methyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
3-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-5-methyl-1H-indole-2-carboxylic acid