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3-[2-(3-fluorophenyl)-3-oxopiperazin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
2-methyl-6-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-{[7-(2-methoxy-2-phenylacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-6-methoxypyrimidin-4-amine
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-6-methylpyridine-3-carboxamide
3-{2-[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)-3-phenylpyrrolidine-2,5-dione
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
2,6-dihydroxy-N-[2-(1H-indol-1-yl)ethyl]-N-methylbenzamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(trimethylpyrimidin-4-yl)piperidin-3-yl]propanoic acid
methyl 2-(diethylsulfamoyl)-6-(3-methylbutyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl (1R,3S,3aR,6aS)-3-(furan-3-yl)-1-(3-methoxy-3-oxopropyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-(morpholin-3-yl)ethan-1-one
4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-1-(1H-indazol-6-yl)-5-methylpiperazin-2-one
2-(3-methyl-1,2-oxazol-5-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl]methanol
N,2-dimethyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl 5-chloro-3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-sulfonyl}thiophene-2-carboxylate
(3R,4R)-1-(2H-1,3-benzodioxol-4-ylmethyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
6-{4-[(dimethylamino)methyl]phenyl}-2-methylquinoline-4-carboxylic acid
2-(ethylsulfanyl)-5-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)pyrimidine
1-[4-(4-methylbenzenesulfonyl)piperazin-1-yl]-3-(pyrazin-2-yl)propan-1-one
1-cyclohexyl-4-[6-(pyridin-3-yl)pyridine-3-carbonyl]-1,4-diazepane
6-(2,3-dihydro-1H-isoindol-2-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-(1-{[1-(2-ethylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(2-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1H-pyrrol-1-yl)pyridine
4-(2-methoxyphenoxy)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methoxyethoxy)ethan-1-one
3-{[1-(2-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
3-{[2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}(propyl)amino)ethan-1-ol
N-(propan-2-yl)-1-[(1s,4s)-4-[3-(pyridin-3-yl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
7-(4-methylphenyl)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}oxolane-3-carboxamide
3-[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
N-cyclobutyl-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2,6-dimethyl-5-{2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]but-3-en-1-one
3-[(4aR,7aS)-6,6-dioxo-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-cyclopropyl-N-propylacetamide
(3S,4S)-3-hydroxy-4-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-N-(2-methylphenyl)pyrrolidine-1-carboxamide
5-{1-[(3-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
2-(dimethylamino)-7-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
1-{[1-(2-fluorophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide