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2-{3-[3-(dimethylamino)propoxy]phenyl}-1H-1,3-benzodiazole-6-carboxylic acid
1-ethyl-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
5-(2-chlorophenyl)-N-[2-(propane-2-sulfonyl)ethyl]furan-2-carboxamide
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(4-chloro-1H-pyrazol-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]ethan-1-one
4-[7-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
[(3R,5R)-1-(3-phenyl-1,2-oxazole-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
8-(2-ethoxyacetyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
4-[(2H-1,3-benzodioxol-4-ylmethyl)amino]-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
5-(dimethylamino)-2-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
4-(2-methoxyphenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-(cyclohexylmethyl)-3-hydroxy-3-({[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)piperidin-2-one
(4aS,8aR)-6-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-[3-cyclopentyl-5-(4-sulfamoylphenyl)-1H-1,2,4-triazol-1-yl]acetic acid
(3aR,5R,6S,7aS)-2-(1-benzylpiperidin-4-yl)-octahydro-1H-isoindole-5,6-diol
5-methyl-14-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-ethyl-6-(6-fluoroquinolin-8-yl)pyridine-3-carboxamide
1-(2-chlorophenyl)-3-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}urea
N-[2-(3,4-dimethylphenyl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
2-[4-(9H-fluoren-2-ylmethyl)morpholin-3-yl]acetic acid
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]propanamide
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-[4-(trifluoromethyl)benzoyl]piperidine
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
3-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)-1-(pyrrolidin-1-yl)propan-1-one
(2S,4S)-4-amino-1-[2-(4-ethoxyphenyl)acetyl]-N-methylpyrrolidine-2-carboxamide
1-amino-3-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]propan-2-ol
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-methoxyethan-1-one
5-(propan-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2-oxazole-3-carboxamide
N-methyl-4-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
N-methyl-N-[2-(oxan-2-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
4-(2-methyl-1H-imidazol-1-yl)-1-(quinolin-2-ylmethyl)piperidine-4-carboxylic acid
6-fluoro-4-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
2-[4-(5-methoxy-1H-indole-2-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-({3-methyl-7-[4-(2-oxopyrrolidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,3-dihydroxypropyl)-1,3-oxazole-4-carboxamide
N-{4-[ethyl(phenyl)carbamoyl]phenyl}-3-(hydroxymethyl)morpholine-4-carboxamide
1-methyl-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-{3-[3-(3-ethylphenoxy)azetidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-methyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]furan-2-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(oxan-4-yl)-decahydro-1,6-naphthyridin-2-one
N-[2-(dimethylamino)-1-phenylethyl]-8-fluoro-N-methylquinoline-2-carboxamide