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N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-3-(2-methylphenyl)benzamide
1-ethyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-N,2,2-trimethyloxan-4-amine
N-[(3,5-dichloro-2-methoxyphenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-(4-oxo-4H-chromen-6-yl)urea
3-fluoro-4-{4-[1-(morpholin-4-yl)ethyl]phenyl}benzene-1-sulfonamide
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
1-benzyl-8-(butan-2-yl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazine-1-carboxamide
6-(cyclopropylamino)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
dimethyl[3-(2-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
3-(1-butyl-1H-imidazol-2-yl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
5-(3,6-dimethylpyrazin-2-yl)thiophene-2-carboxylic acid
5-{1-[(3-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(4-methoxyphenyl)-1-benzofuran-2-carboxamide
3-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
3-(3,6-dimethylpyrazin-2-yl)-9-methyl-3,9-diazaspiro[5.6]dodecane
4-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}morpholine
4-[(2S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carbonyl]morpholine
6-methyl-2-{2-[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-(1,3-dihydroxypropan-2-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-2,7-diazaspiro[4.5]decane
N-cycloheptyl-2-cyclopropyl-N-[(3-methoxyphenyl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[(3-methylthiophen-2-yl)methyl]propanamide
3-{[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)oxy]methyl}pyridine
N-benzyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-methyl-3-[3-(1H-pyrazol-3-yl)phenyl]benzamide
N-cyclohexyl-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
1-[4-(1H-pyrazol-5-yl)phenyl]-3-(2,2,6,6-tetramethylpiperidin-4-yl)urea
5-ethyl-1'-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2S,4S)-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-cyclopentaneamido-1-methylpyrrolidine-2-carboxamide
5-[3-(1H-pyrazol-3-yl)phenyl]pyridin-2-amine
4-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)(pyridin-3-yl)methyl]morpholine
2-[(5-ethylpyrimidin-2-yl)amino]-N,N-dimethylethane-1-sulfonamide
N-{1-[1-(cyclohexylmethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-2-methylpropyl}acetamide
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
3-[2-(2,4-dimethoxyphenyl)-1H-imidazol-1-yl]piperidin-2-one
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-(4-methyl-3-phenyl-1H-pyrazol-1-yl)acetamide
1-(2-fluorophenyl)-5-[1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(2-methylpropyl)-1H-1,2,4-triazole
4-({3-[3-(6-methylpyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}methyl)benzonitrile
(1S,5R)-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-fluorophenoxy)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]ethan-1-one
9-[(5-ethylpyridin-2-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
3-[(2-fluorophenyl)methyl]-4-[(2-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-6-(4-chloro-2-fluorobenzoyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-(1,3-benzothiazole-6-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-(butan-2-yl)phenoxy]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylacetamide
7-fluoro-N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N4-[(3,5-difluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine