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(3aR,6aR)-2-(6-ethyl-5-fluoropyrimidin-4-yl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)piperidin-2-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(2-methyl-1H-imidazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
5-[(1R,4R)-bicyclo[2.2.1]hept-5-en-2-yl]-3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazole
N-{2-[1-(2-hydroxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}-2-(thiophen-2-yl)acetamide
2-methyl-4-[2-(4-phenylpiperidin-1-yl)ethyl]-1-(propan-2-yl)piperazine
1-(4-{[(2R)-oxolan-2-ylmethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-[4-(1,3-benzoxazol-2-yl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
7-(cyclopropylmethyl)-2-[(2-propylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-4-amino-N-methyl-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidine-2-carboxamide
1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-methoxypiperidine
5-[(3-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-(prop-2-en-1-yl)imidazolidine-2,4-dione
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3-(4-methylphenoxymethyl)piperidine
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-oxopyrrolidin-1-yl)acetamide
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(1-methoxypropan-2-yl)piperidine
(1S,5R)-3-[3-(2-chlorophenyl)propanoyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(piperidin-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[2-(pyridin-3-yl)acetyl]piperidine-3-carboxylate
3-[2-(3-methoxyphenyl)ethyl]-N,N-dimethylpiperidine-1-sulfonamide
N-[(3R,4R)-1-(3,6-dimethylpyrazin-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
2-[3-fluoro-5-(trifluoromethyl)phenyl]-4-(piperidine-1-carbonyl)pyridine
2-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinoxaline
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
1-[2-(adamantan-1-yl)acetyl]imidazolidin-4-one
[(4-fluorophenyl)methyl](methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
(4aS,8aR)-6-phenylmethanesulfonyl-1-propyl-decahydro-1,6-naphthyridin-2-one
(cyclohexylmethyl)(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
1-methyl-9-{[2-(2-phenylethynyl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
3-{[(3-methyl-1,2-oxazol-5-yl)methyl]sulfamoyl}-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
5-(2-methylpropyl)-1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]propanamide
7-oxo-N-[phenyl(pyridin-4-yl)methyl]-2-(2-phenylacetamido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-methyl-2-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-1,3-benzodiazole
8-(4-chloro-3-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(3-acetamidopropanoyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-(4-fluorophenoxy)-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
1-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}urea
1-(pyrimidin-2-yl)-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4-diazepane
5-methoxy-2-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyran-4-one
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-(4-fluorophenyl)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-methanesulfonamidoethyl)acetamide
(1R,2R,6S,7S)-4-(pyridin-4-yl)-4-azatricyclo[5.2.1.02,6]decane
3-[(dimethylamino)methyl]-1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
2,5-dimethyl-3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
1-{1-[2-(phenylsulfanyl)ethyl]piperidin-4-yl}piperidin-3-ol